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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLCB3 1-(1,3-Benzodioxol-5-yl)-3-o-cumenyl-urea NA 122542 NA NA NA NA BindingDB
PLCB3 2-[[4-[(5E)-5-(2-furanylmethylidene)-4-oxo-2-sulfanylidene-3-thiazolidinyl]-1-oxobutyl]amino]-5-hydroxybenzoic acid NA 122465 NA NA NA NA BindingDB
PLCB3 2-[2-(methylanilino)-2-oxoethoxy]-N-(2-phenoxyethyl)benzamide NA 122435 NA NA NA NA BindingDB
PLCB3 (Z)-2-(4-ethylbenzylidene)-6-hydroxy-7-((4-(2-hydroxyethyl)piperazin-1-yl)methyl)benzofuran-3(2H)-one NA 122491 NA NA NA NA BindingDB
PLCB3 4-[3-(5-Furan-2-yl-2H-pyrazol-3-yl)-5-mercapto-[1,2,4]triazol-4-yl]-benzoic acid NA 122493 NA NA NA NA BindingDB
PLCB3 3-(2,4-Dichlorobenzyl)-5-methoxy-1-methyl-pyrido[2,3-d]pyrimidine-2,4-quinone NA 122483 NA NA NA NA BindingDB
PLCB3 3-[5-[(E)-(1-oxo-[1,3]thiazolo[3,2-a]benzimidazol-2-ylidene)methyl]furan-2-yl]benzoic acid NA 122487 NA NA NA NA BindingDB
PLCB3 4-[(5Z)-5-[(E)-3-(furan-2-yl)prop-2-enylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]butanoic acid NA 122481 NA NA NA NA BindingDB
PLCB3 4-tert-butyl-N-phenylcyclohexane-1-carboxamide NA 122440 NA NA NA NA BindingDB
PLCB3 1-(2,3-Dihydroindol-1-yl)-2-(1-methylindol-3-yl)sulfonylethanone NA 122493 NA NA NA NA BindingDB
PLCB3 3-{1,3-dioxo-5-[(3,4,5-trimethoxybenzoyl)amino]-1,3-dihydro-2H-isoindol-2-yl}propanoic acid NA 122467 NA NA NA NA BindingDB
PLCB3 3-(3,5-Dichloroanilino)-1-thiophen-2-ylpropan-1-one NA 122542 NA NA NA NA BindingDB
PLCB3 3-(4-methylphenyl)sulfonyl-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)propanamide NA 122452 NA NA NA NA BindingDB
PLCB3 3-(4-Bromo-2-chloro-phenoxy)propyl-(2-methoxyethyl)amine;oxalic acid NA 122506 NA NA NA NA BindingDB
PLCB3 bis[2-[2-(1H-indol-3-yl)ethylamino]-2-oxoethyl] benzene-1,2-dicarboxylate NA 122579 NA NA NA NA BindingDB
PLCB3 7-Amino-6-chloro-5,8-dioxonaphthalene-2-sulfonamide NA 122373 NA NA NA NA BindingDB
PLCB3 3-[4-(Azepan-1-yl)-3-nitro-phenyl]-3-(2-naphthalen-1-ylethanoylamino)propanamide NA 122481 NA NA NA NA BindingDB
PLCB3 3-[4-(3-chlorophenyl)piperazino]sulfonyl-5-nitro-1H-indole NA 122481 NA NA NA NA BindingDB
PLCB3 [3-[4-(4-Fluorophenyl)piperazino]sulfonylphenyl]-[3-(trifluoromethyl)piperidino]methanone NA 122478 NA NA NA NA BindingDB
PLCB3 [2-[(6-Amino-1-benzyl-2,4-dioxopyrimidin-5-yl)-ethylamino]-2-oxoethyl] 4-formylbenzoate NA 122492 NA NA NA NA BindingDB