| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLAU |
|
NA |
236000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
3-[(2-Methylpropan-2-yl)oxycarbonylamino]propyl 3,4,5-trihydroxybenzoate |
NA |
188700 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
3-hydroxy-N-(3-hydroxyphenyl)sulfonyl-N-octylbenzenesulfonamide |
NA |
100300 |
NA |
NA |
NA |
NA |
BindingDB |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-7-methyl-6-[(3-methyl-2,5-dioxoimidazolidin-1-yl)methyl]pyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-(4-fluorophenyl)-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-(4-methoxyphenyl)-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-3-(4-propylphenyl)imidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-3-(4-sulfamoylphenyl)imidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-(4-carbamoylphenyl)-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-(4-cyanophenyl)-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-3-(3-sulfamoylphenyl)imidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-(3-carbamoylphenyl)-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-(3-cyanophenyl)-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-3-[4-(2-oxopropoxy)phenyl]imidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-[4-(2-amino-2-oxoethoxy)phenyl]-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-[4-(cyanomethoxy)phenyl]-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-[4-(4-methoxyphenoxy)phenyl]-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-3-[4-(pyridin-4-ylmethoxy)phenyl]imidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-3-(4-quinolin-6-yloxyphenyl)imidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| PLAU |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-[4-(2-carbamoylphenoxy)phenyl]-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |