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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLAU (R)-N-[(5-chloro-2-ethyl-benzylcarbamoyl)-methyl]-4-(1-oxy-pyridin-2-yl)-2-phenylmethanesulfonylamino-butyramide 150000 NA NA NA NA NA BindingDB|TTD
PLAU [Amino(phenyl)methylidene]azanium 180000|380000 NA NA NA NA NA BindingDB
PLAU 3-Amino-N-{3-[(S)-2-[4-(2-amino-ethyl)-piperidin-1-yl]-1-(3-aminomethyl-benzyl)-2-oxo-ethylsulfamoyl]-phenyl}-propionamide 1000000 NA NA NA NA NA TTD
PLAU 3-Amino-N-{3-[(S)-2-[4-(2-amino-ethyl)-piperidin-1-yl]-1-(4-aminomethyl-benzyl)-2-oxo-ethylsulfamoyl]-phenyl}-propionamide 1000000 NA NA NA NA NA TTD
PLAU US8569313, Inhibitor 35 129000 NA NA NA NA NA BindingDB|TTD
PLAU methyl (2S)-1-[(2S)-2-[[3-(3-aminopropanoylamino)phenyl]sulfonylamino]-3-(3-carbamimidoylphenyl)propanoyl]piperidine-2-carboxylate 126000 NA NA NA NA NA BindingDB|TTD
PLAU (2S)-1-[(2S)-2-[[3-(3-aminopropanoylamino)phenyl]sulfonylamino]-3-(3-carbamimidoylphenyl)propanoyl]piperidine-2-carboxylic acid 193000 NA NA NA NA NA BindingDB|TTD
PLAU [4-(4-Aminobutyl)-3,6,9-trioxo-2,5,8-triazabicyclo[8.3.1]tetradeca-1(14),10,12-trien-11-yl]methyl-methyl-phenylsulfanium;bromide 500000 NA NA NA NA NA TTD
PLAU Cyanopeptolin 1020 NA 605000 NA NA NA NA TTD
PLAU 3-[2-Amino-3-(4-methyl-piperidin-1-yl)-3-oxo-propyl]-benzamidine 800000 NA NA NA NA NA BindingDB|TTD
PLAU N-(4-fluorobenzyl)-2-hydrazinyl-2-oxoacetamide NA 478000|649000|1251500 NA NA NA NA BindingDB
PLAU N-[3-(trifluoromethyl)phenyl]guanidine 418794|419000|418793.57 NA NA NA NA NA BindingDB|TTD
PLAU N-Hexyl-2-hydrazineyl-2-oxoacetamide NA 1208000|2097000|3839000 NA NA NA NA BindingDB
PLAU Tranexamic acid 2000000 NA NA NA NA NA BindingDB|PubChem|TTD
PLAU Vaborbactam NA 1000000 NA NA NA NA PubChem|TTD
PLAU 4-amino-5-chloro-N-(diaminomethylidene)-2-methoxybenzamide NA 222000 NA NA NA NA TTD
PLAU 5,6-dichloro-N-(diaminomethylidene)pyridine-3-carboxamide NA 1000000 NA NA NA NA BindingDB|TTD
PLAU 3-amino-N-(diaminomethylidene)-5-(2-phenylethylamino)pyrazine-2-carboxamide NA 120000 NA NA NA NA BindingDB|TTD
PLAU 2-[[6-Amino-3-chloro-5-(diaminomethylidenecarbamoyl)pyrazin-2-yl]amino]ethyl-ethoxyphosphinic acid NA 1000000 NA NA NA NA TTD
PLAU 3-[[6-Amino-3-chloro-5-(diaminomethylidenecarbamoyl)pyrazin-2-yl]amino]propanoic acid NA 102000 NA NA NA NA BindingDB|TTD