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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLAT 3-Hydroxy-4-methoxy-anthracene-2-carboxylic acid (6-guanidino-pyridin-3-yl)-amide 150000 NA NA NA NA NA BindingDB|TTD
PLAT 3-Hydroxy-4-iodo-anthracene-2-carboxylic acid (6-guanidino-pyridin-3-yl)-amide 225000 NA NA NA NA NA BindingDB|TTD
PLAT 4-Bromo-3-hydroxy-anthracene-2-carboxylic acid (6-guanidino-pyridin-3-yl)-amide 506000 NA NA NA NA NA BindingDB|TTD
PLAT 3-Hydroxy-anthracene-2-carboxylic acid (6-guanidino-pyridin-3-yl)-amide 338000 NA NA NA NA NA BindingDB|TTD
PLAT 3-Hydroxy-4-methoxy-anthracene-2-carboxylic acid (4-guanidino-phenyl)-amide 181000 NA NA NA NA NA BindingDB|TTD
PLAT N-(4-Guanidino-phenyl)-2-hydroxy-3-iodo-5-methyl-benzamide 563000 NA NA NA NA NA TTD
PLAT 3-Bromo-N-(4-guanidino-phenyl)-2-hydroxy-5-methyl-benzamide 258000 NA NA NA NA NA BindingDB|TTD
PLAT 113000 NA NA NA NA NA BindingDB
PLAT 3-Carbamimidoyl-N-[(R)-phenyl-(2''-sulfamoyl-biphenyl-4-ylcarbamoyl)-methyl]-benzamide NA 180000 NA NA NA NA TTD
PLAT (3S)-2-(3-carbamimidoylbenzoyl)-N-[4-(2-sulfamoylphenyl)phenyl]-3,4-dihydro-1H-isoquinoline-3-carboxamide NA 180000 NA NA NA NA BindingDB|TTD
PLAT H-Tic-Pro-Arg-al NA 430000 NA NA NA NA BindingDB|TTD
PLAT 3-[(R)-3-(4-Methanesulfonyl-piperazin-1-yl)-3-oxo-2-(2,2,5,7,8-pentamethyl-chroman-6-sulfonylamino)-propyl]-benzamidine 470000 NA NA NA NA NA BindingDB|TTD
PLAT N-(5-Phenyl-isoquinolin-1-yl)-guanidine 123900 NA NA NA NA NA BindingDB|TTD
PLAT N-(4-Chloro-isoquinolin-1-yl)-guanidine 128500 NA NA NA NA NA BindingDB|TTD
PLAT N-(4-Bromo-isoquinolin-1-yl)-guanidine 159200 NA NA NA NA NA BindingDB|TTD
PLAT N-(5-Bromo-isoquinolin-1-yl)-guanidine 140100 NA NA NA NA NA BindingDB|TTD
PLAT N-(7-Phenyl-isoquinolin-1-yl)-guanidine 123900 NA NA NA NA NA BindingDB|TTD
PLAT (S)-1-(3-Phenyl-3-pyridin-4-yl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA 436000 NA NA NA NA NA BindingDB|TTD
PLAT (S)-1-(3-Phenyl-3-pyridin-3-yl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA 746000 NA NA NA NA NA BindingDB|TTD
PLAT (S)-1-(3-Phenyl-3-pyridin-2-yl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA 1000000 NA NA NA NA NA TTD