| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLCB3 |
|
NA |
122476 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
|
NA |
122457 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
2-[(2R,4aS,12aS)-8-[(2-fluorophenyl)carbamoylamino]-5-methyl-6-oxidanylidene-2,3,4,4a,12,12a-hexahydropyrano[2,3-c][1,5]benzoxazocin-2-yl]-N-[(4-phenylphenyl)methyl]ethanamide |
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
methyl 2-[(2S,4aR,12aR)-8-[(3-fluorophenyl)carbonylamino]-5-methyl-6-oxidanylidene-2,3,4,4a,12,12a-hexahydropyrano[2,3-c][1,5]benzoxazocin-2-yl]ethanoate |
NA |
122430 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
|
NA |
122562 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
Methacycline hydrochloride |
NA |
122490 |
NA |
NA |
NA |
NA |
PubChem |
| PLCB3 |
|
NA |
122387 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
pyrazinic acid [(1S,2R,3S)-1''-benzyl-2-(hydrocinnamoylamino)-2''-keto-spiro[cyclohexane-3,3''-indoline]-1-yl] ester |
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
|
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
2-[(5Z)-5-[(E)-3-(furan-2-yl)prop-2-enylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]butanedioic acid |
NA |
122454 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
dimethyl 2-[(3R,6S)-1-acetyl-6-[(4-methylphenyl)sulfonylcarbamoyl]-3,6-dihydro-2H-pyridin-3-yl]propanedioate |
NA |
122459 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
(3S,6S)-1-acetyl-3-ethyl-N-tosyl-3,6-dihydro-2H-pyridine-6-carboxamide |
NA |
122467 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
(3R,6S)-1-acetyl-3-(1H-indol-3-yl)-N-tosyl-3,6-dihydro-2H-pyridine-6-carboxamide |
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
4-[(E)-[3-(2-methylanilino)-4-oxonaphthalen-1-ylidene]amino]sulfonylbenzoic acid |
NA |
122481 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
Adenosine Phosphate |
NA |
122473 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
3-[2-[(E)-[1-(4-chlorophenyl)-2,5-dioxoimidazolidin-4-ylidene]methyl]pyrrol-1-yl]benzoic acid |
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
AC1Lde0K |
NA |
101771 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
5-[[2-[(5Z)-5-(furan-2-ylmethylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetyl]amino]-2-hydroxybenzoic acid |
NA |
122481 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
4-({[(5Z)-5-(furan-2-ylmethylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetyl}amino)-2-hydroxybenzoic acid |
NA |
122451 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCB3 |
(Z)-5-((E)-3-(furan-2-yl)allylidene)-3-(4-hydroxyphenyl)-2-thioxothiazolidin-4-one |
NA |
122562 |
NA |
NA |
NA |
NA |
BindingDB |