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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLCB3 (2-Methoxyphenyl)methyl 3-pyrrolidin-1-ylsulfonylbenzoate NA 122506 NA NA NA NA BindingDB
PLCB3 N,N''-bis(4-keto-2-thioxo-thiazolidin-3-yl)oxamide NA 122457 NA NA NA NA BindingDB
PLCB3 3-nitro-4-[2-[(E)-(2-oxidanyl-4-oxidanylidene-cyclohexa-2,5-dien-1-ylidene)methyl]hydrazinyl]benzenesulfonamide NA 122506 NA NA NA NA BindingDB
PLCB3 Alpha,beta-methylene adenosine 5'-diphosphate NA 122493 NA NA NA NA BindingDB
PLCB3 4-[[(E)-3-(furan-2-yl)prop-2-enoyl]carbamothioylamino]benzoic acid NA 122476 NA NA NA NA BindingDB
PLCB3 4-{(E)-[2-(3-hydroxybenzoyl)hydrazono]methyl}phenyl benzoate NA 122480 NA NA NA NA BindingDB
PLCB3 2-(3,4-dichlorophenyl)-N'-[(2-thienylcarbonyl)oxy]ethanimidamide NA 122471 NA NA NA NA BindingDB
PLCG1 2-(1,5-Dimethyl-3-oxo-2-phenylpyrazol-4-yl)benzo[de]isoquinoline-1,3-dione NA 122493 NA NA NA NA BindingDB
PLCG1 6-{[cyclohexyl(methyl)amino]methyl}-N-(2-ethoxyphenyl)-1,3,5-triazine-2,4-diamine NA 122517 NA NA NA NA BindingDB
PLCG1 N-(4-benzamido-3-methylphenyl)-1,3-benzodioxole-5-carboxamide NA 122480 NA NA NA NA BindingDB
PLCG1 N-(4-Benzoylamino-3-methyl-phenyl)-3-ethoxy-benzamide NA 122382 NA NA NA NA BindingDB
PLCG1 N-[2-chloro-4-[(4-propan-2-yloxybenzoyl)amino]phenyl]furan-2-carboxamide NA 122498 NA NA NA NA BindingDB
PLCG1 (2E)-3-{1-[3-(dipropylamino)-2-hydroxypropyl]-1H-indol-3-yl}-1-thien-2-ylprop-2-en-1-one NA 122460 NA NA NA NA BindingDB
PLCG1 3-(2-methoxyphenyl)-2-{[(tetrahydro-2-furanylmethyl)amino]methyl}-4(3H)-quinazolinone NA 122382 NA NA NA NA BindingDB
PLCG1 4-(5-(Furan-2-ylmethylene)-4-oxo-2-thioxothiazolidin-3-yl)butanoic acid NA 122506 NA NA NA NA BindingDB
PLCG1 N-[1-(1-Cyclopentyl-1H-tetrazol-5-ylmethyl)-piperidin-4-yl]-2-methyl-benzamide NA 122493 NA NA NA NA BindingDB
PLCG1 N-(6-benzamido-4-methylpyridin-3-yl)thiophene-2-carboxamide NA 122469 NA NA NA NA BindingDB
PLCG1 N-(4-methoxyphenyl)-3-(2-thienyl)-6-(trifluoromethyl)thieno[3,2-b]pyridine-2-carboxamide NA 122457 NA NA NA NA BindingDB
PLCG1 5-(4-chlorophenyl)-1-phenyl-1H-pyrazol-4-yl phenyl sulfone NA 122478 NA NA NA NA BindingDB
PLCG1 5-(4-fluorophenyl)-1-phenyl-1H-pyrazol-4-yl phenyl sulfone NA 122506 NA NA NA NA BindingDB