| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLCG1 |
N-[4-[(2,6-dimethoxypyrimidin-4-yl)sulfamoyl]phenyl]-2-(1,3-dioxoisoindol-2-yl)acetamide |
NA |
122387 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
(5Z)-5-(furan-2-ylmethylidene)-3-pyridin-3-yl-2-sulfanylidene-1,3-thiazolidin-4-one |
NA |
122443 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
3-[4-[(5Z)-5-(furan-2-ylmethylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]butanoylamino]benzoic acid |
NA |
122499 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
2,4-Dinitropyrimidinyl-2-thiophenol |
NA |
122702 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
Methyl 2-[2-[(4-tert-butylbenzoyl)amino]propanoylamino]-3-(4-hydroxyphenyl)propanoate |
NA |
122508 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
2-(2,5-diketospiro[imidazolidine-4,1''-tetralin]-1-yl)-N-homoveratryl-N-methyl-acetamide |
NA |
122490 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
1-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)-3-[(E)-[(E)-3-(4-nitrophenyl)prop-2-enylidene]amino]thiourea |
NA |
122506 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
(E)-4-(3-(5-(furan-2-ylmethylene)-4-oxo-2-thioxothiazolidin-3-yl)propanamido)-2-hydroxybenzoic acid |
NA |
122481 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
1-(1,3-Benzodioxol-5-yl)-3-o-cumenyl-urea |
NA |
122542 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
2-[[4-[(5E)-5-(2-furanylmethylidene)-4-oxo-2-sulfanylidene-3-thiazolidinyl]-1-oxobutyl]amino]-5-hydroxybenzoic acid |
NA |
122465 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
2-[2-(methylanilino)-2-oxoethoxy]-N-(2-phenoxyethyl)benzamide |
NA |
122435 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
(Z)-2-(4-ethylbenzylidene)-6-hydroxy-7-((4-(2-hydroxyethyl)piperazin-1-yl)methyl)benzofuran-3(2H)-one |
NA |
122491 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
4-[3-(5-Furan-2-yl-2H-pyrazol-3-yl)-5-mercapto-[1,2,4]triazol-4-yl]-benzoic acid |
NA |
101799 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
3-(2,4-Dichlorobenzyl)-5-methoxy-1-methyl-pyrido[2,3-d]pyrimidine-2,4-quinone |
NA |
122483 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
3-[5-[(E)-(1-oxo-[1,3]thiazolo[3,2-a]benzimidazol-2-ylidene)methyl]furan-2-yl]benzoic acid |
NA |
122487 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
4-[(5Z)-5-[(E)-3-(furan-2-yl)prop-2-enylidene]-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]butanoic acid |
NA |
122481 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
4-tert-butyl-N-phenylcyclohexane-1-carboxamide |
NA |
122440 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
1-(2,3-Dihydroindol-1-yl)-2-(1-methylindol-3-yl)sulfonylethanone |
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
3-{1,3-dioxo-5-[(3,4,5-trimethoxybenzoyl)amino]-1,3-dihydro-2H-isoindol-2-yl}propanoic acid |
NA |
122467 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
3-(3,5-Dichloroanilino)-1-thiophen-2-ylpropan-1-one |
NA |
122542 |
NA |
NA |
NA |
NA |
BindingDB |