| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLCG1 |
N,5-bis(3,4-dimethoxyphenyl)isoxazole-3-carboxamide |
NA |
122527 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
ethyl (2Z)-cyano(1-methylpyrimidin-4(1H)-ylidene)acetate |
NA |
122567 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
4-amino-N-cyclohexyl-2-methylsulfanyl-1,3-thiazole-5-carboxamide |
NA |
122542 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-isobutyl-2-[(5-methyl-3-thienyl)carbonyl]hydrazinecarbothioamide |
NA |
122473 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-[3-[4-(2-fluorophenyl)piperazin-1-yl]-1,4-dioxonaphthalen-2-yl]-4-methylbenzenesulfonamide |
NA |
122475 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
2-(4-Chlorophenyl)sulfonylquinoxaline |
NA |
122579 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
10-(Diiodomethylidene)phenanthren-9-one |
NA |
122481 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
Methyl 1-[(4-bromo-2-chlorophenoxy)acetyl]-2-pyrrolidinecarboxylate |
NA |
122483 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-[4-(phenoxymethyl)-2-thiazolyl]-1-adamantanecarboxamide |
NA |
122505 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
3-(2,4-dichlorophenyl)-1H-quinazoline-2,4-dione |
NA |
122403 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-butyl-2-[(5-ethyl-3-thienyl)carbonyl]hydrazinecarbothioamide |
NA |
122355 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-[4-(5-tert-butyltriazol-1-yl)phenyl]-3-methoxybenzamide |
NA |
122411 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-(4-(4-Acetamidophenyl)thiazol-2-yl)-1-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)-5-oxopyrrolidine-3-carboxamide |
NA |
122517 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-(2-chlorophenyl)-2-[(3-chlorophenyl)sulfinyl]acetamide |
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
(2E,4S,4aR,5S,5aR,12aS)-2-[azanyl(oxidanyl)methylidene]-4-(dimethylamino)-6-methylidene-5,10,11,12a-tetrakis(oxidanyl)-4,4a,5,5a-tetrahydrotetracene-1,3,12-trione;hydrochloride |
NA |
122490 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
ML228 Analog |
NA |
122380 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-[(2-methoxynaphthalen-1-yl)methyl]-2-(4-methoxyphenyl)ethanamine |
NA |
122506 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-[2-[1-[2-(4-methylphenoxy)ethyl]-2-benzimidazolyl]ethyl]cycloheptanecarboxamide |
NA |
122506 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-(4-chlorophenyl)-N'-hydroxybenzenecarboximidamide |
NA |
122433 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
3-[1-[1-(1-cyclohexyltetrazol-5-yl)propyl]-4-piperidyl]-1H-benzimidazol-2-one |
NA |
122480 |
NA |
NA |
NA |
NA |
BindingDB |