| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLCG1 |
2-[3-butyl-8-(hydroxymethyl)-2,6-dioxo-7-propylpurin-1-yl]-N-(3-chloro-4-methoxyphenyl)acetamide |
NA |
122506 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-butyl-2-[(5-methyl-3-thienyl)carbonyl]hydrazinecarbothioamide |
NA |
122464 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
Ethyl 2-[[4-(2-methylphenyl)-5-[(2-oxo-1,3-benzothiazol-3-yl)methyl]-1,2,4-triazol-3-yl]sulfanyl]acetate |
NA |
122451 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
(5Z)-5-[(2E)-3-(5-nitro-2-furyl)prop-2-enylidene]-2-thioxo-1,3-thiazolidin-4-one |
NA |
122468 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
I-OMe-Tyrphostin AG 538 |
NA |
122486 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
|
NA |
107767 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
(E)-2-cyano-3-(3,4,5-trihydroxyphenyl)prop-2-enamide |
NA |
122371 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
|
NA |
122481 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
|
NA |
122476 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
|
NA |
122457 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
2-[(2R,4aS,12aS)-8-[(2-fluorophenyl)carbamoylamino]-5-methyl-6-oxidanylidene-2,3,4,4a,12,12a-hexahydropyrano[2,3-c][1,5]benzoxazocin-2-yl]-N-[(4-phenylphenyl)methyl]ethanamide |
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
methyl 2-[(2S,4aR,12aR)-8-[(3-fluorophenyl)carbonylamino]-5-methyl-6-oxidanylidene-2,3,4,4a,12,12a-hexahydropyrano[2,3-c][1,5]benzoxazocin-2-yl]ethanoate |
NA |
122430 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
|
NA |
122562 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
Methacycline hydrochloride |
NA |
122490 |
NA |
NA |
NA |
NA |
PubChem |
| PLCG1 |
|
NA |
122387 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
pyrazinic acid [(1S,2R,3S)-1''-benzyl-2-(hydrocinnamoylamino)-2''-keto-spiro[cyclohexane-3,3''-indoline]-1-yl] ester |
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
|
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
(3S,6S)-1-acetyl-3-ethyl-N-tosyl-3,6-dihydro-2H-pyridine-6-carboxamide |
NA |
122467 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
3-[2-[(E)-[1-(4-chlorophenyl)-2,5-dioxoimidazolidin-4-ylidene]methyl]pyrrol-1-yl]benzoic acid |
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
5-[[2-[(5Z)-5-(furan-2-ylmethylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]acetyl]amino]-2-hydroxybenzoic acid |
NA |
122481 |
NA |
NA |
NA |
NA |
BindingDB |