| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLCG1 |
4-({[(5Z)-5-(furan-2-ylmethylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]acetyl}amino)-2-hydroxybenzoic acid |
NA |
122451 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
(Z)-5-((E)-3-(furan-2-yl)allylidene)-3-(4-hydroxyphenyl)-2-thioxothiazolidin-4-one |
NA |
122562 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
2-((Z)-5-((E)-3-(furan-2-yl)allylidene)-4-oxo-2-thioxothiazolidin-3-yl)propanoic acid |
NA |
122491 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
|
NA |
122469 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
|
NA |
122464 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
5-[2-[(5Z)-5-(furan-2-ylmethylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]propanoylamino]-2-hydroxybenzoic acid |
NA |
122457 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
3-(2-morpholin-4-ylethyl)-5H-pyrimido[5,4-b]indol-4-one |
NA |
122453 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
Methyl 2-[(5-cyano-3,3,8-trimethyl-1,4-dihydropyrano[3,4-c]pyridin-6-yl)oxy]acetate |
NA |
122521 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-1-Naphthylbenzamide |
NA |
122537 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
|
NA |
122502 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
(2Z)-2-[(5-methylfuran-2-yl)methylidene]-1,3-dioxoindene-5-carboxylic acid |
NA |
122490 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
N-(3-chlorophenyl)-2-(3-ethyl-5-methyl-7-oxo-2-sulfanylidene-[1,3]thiazolo[4,5-d]pyrimidin-6-yl)acetamide |
NA |
122493 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
3,5-Bisnitro-4-methyl-2-(phenylsulfanyl)pyridine |
NA |
122449 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
3-[3-(3-Furan-2-yl-acryloyl)-thioureido]-benzoic acid |
NA |
122422 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
2-(benzylthio)-N-(3-fluorophenyl)acetamide |
NA |
122432 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
(2-Methoxyphenyl)methyl 3-pyrrolidin-1-ylsulfonylbenzoate |
NA |
122506 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
3-nitro-4-[2-[(E)-(2-oxidanyl-4-oxidanylidene-cyclohexa-2,5-dien-1-ylidene)methyl]hydrazinyl]benzenesulfonamide |
NA |
122506 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
4-[[(E)-3-(furan-2-yl)prop-2-enoyl]carbamothioylamino]benzoic acid |
NA |
122476 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
4-{(E)-[2-(3-hydroxybenzoyl)hydrazono]methyl}phenyl benzoate |
NA |
122480 |
NA |
NA |
NA |
NA |
BindingDB |
| PLCG1 |
2-(3,4-dichlorophenyl)-N'-[(2-thienylcarbonyl)oxy]ethanimidamide |
NA |
122471 |
NA |
NA |
NA |
NA |
BindingDB |