| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLEC |
(3aS,5S,9aS)-2-methyl-5-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]hexahydro-7H-pyrrolo[3,4-g]pyrrolizin-1(2H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(2,6-difluorobenzyl)-5-[(2,6-difluorophenoxy)methyl]isoxazole-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-{4-[(2-Fluorobenzoyl)amino]phenoxy}-2-thiophenecarboxylic acid |
NA |
167613.9|200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-(2-methylphenyl)[1,2,4]triazolo[1,5-c]quinazoline-5(6H)-thione |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-(1,3-dioxoisoindol-2-yl)-N-(4-sulfamoylphenyl)benzamide |
NA |
170750 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-butyl-N-[(6-methoxy-2-oxo-1H-quinolin-3-yl)methyl]-4-methylbenzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
ethyl 2-methyl-4,5-dioxo-4,5-dihydro-3H-benzo[e]indole-1-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-[(1S)-1-(homoveratrylcarbamoyl)-2-methyl-butyl]-1,2-dihydroimidazo[1,2-a]benzimidazole-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
1-[(3-methoxypropyl)amino]-3H-naphtho[1,2,3-de]quinoline-2,7-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
(E)-3-(4-fluorophenyl)-N-[[4-[(6-methoxypyrimidin-4-yl)sulfamoyl]phenyl]carbamothioyl]prop-2-enamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
Methyl 3-[[4-chloro-5-[[(2-chlorobenzoyl)hydrazinylidene]methyl]-2-oxo-1,3-thiazol-3-yl]methyl]benzoate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-[(5-Bromo-furan-2-carbonyl)-amino]-1-butyl-1H-pyrrolo[2,3-b]quinoxaline-3-carboxylic acid ethyl ester |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-[1-butyl-3-(4-methylphenyl)sulfonylpyrrolo[3,2-b]quinoxalin-2-yl]furan-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-[(5Z)-4-oxo-5-[(1-phenyl-3-thiophen-2-ylpyrazol-4-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-3-yl]propanoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-amino-1-benzyl-N-(furan-2-ylmethyl)-1H-pyrrolo[2,3-b]quinoxaline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-Amino-1-phenethyl-1H-pyrrolo[2,3-b]quinoxaline-3-carboxylic acid (furan-2-ylmethyl)-amide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-[1-Butyl-3-(toluene-4-sulfonyl)-1H-pyrrolo[2,3-b]quinoxalin-2-yl]-benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-[3-(benzenesulfonyl)-1-cyclohexyl-2-pyrrolo[3,2-b]quinoxalinyl]benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-[1-Allyl-3-(toluene-4-sulfonyl)-1H-pyrrolo[2,3-b]quinoxalin-2-yl]-benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-amino-N-(furan-2-ylmethyl)-1-(3-methoxypropyl)pyrrolo[3,2-b]quinoxaline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |