| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLEC |
Rhein |
NA |
155815.3|200000|155815 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PLEC |
4-({3-Bromo-4-[(2-fluorobenzyl)oxy]-5-methoxybenzyl}amino)phenol |
NA |
126648.5 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
4,5-Dichloro-2-[oxo-(8-quinolinylamino)methyl]benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(1,3-benzodioxol-5-yl)-5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-Phenylpropanoic acid 2-(dimethylamino)ethyl ester |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(2-furanylmethyl)-2-(4-oxo-5-phenyl-3-thieno[2,3-d]pyrimidinyl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
|
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
methyl 2-[(E)-2-(2-hydroxyphenyl)ethenyl]-1,3,3-trimethylindol-1-ium-5-carboxylate;iodide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-[2-(4-methylphenyl)-2-oxoethoxy]-N-phenylbenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
Ethyl 2-cyano-2-[3-ethyl-5-(1-ethylquinolin-2-ylidene)-4-oxo-1,3-thiazolidin-2-ylidene]acetate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
(5E)-3-benzyl-5-(3-chloro-4-hydroxy-5-methoxybenzylidene)-2-thioxo-1,3-thiazolidin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
[4-[[(3-Fluorobenzoyl)hydrazinylidene]methyl]phenyl] thiophene-2-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
(1-phenyl-1H-1,2,3-triazol-4-yl)methyl N-(4-chlorophenyl)carbamate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2,4-Dibromo-6-[(4-fluoroanilino)methyl]benzenol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(4-chlorophenyl)-4-morpholin-4-ylsulfonylbenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-(4-Carboxybenzyl)-4-(3,5-di-tert-butyl-4-hydroxyphenyl)-2-(phenylamino)-1,3-thiazol-3-ium |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
(5-((3-(4-Isobutoxyphenyl)-1-phenyl-1H-pyrazol-4-YL)methylene)-4-oxo-2-thioxo-1,3-thiazolidin-3-YL)acetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(3,4-dimethoxyphenyl)-2-methyl-1,1-bis(oxidanylidene)-5-thiophen-2-yl-1,2,6-thiadiazine-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-chloro-N-{5-[(4-methylpiperidin-1-yl)sulfonyl]-1,3,4-thiadiazol-2-yl}benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-[2-(4-chlorophenyl)ethyl]-2-(8-methyl-5-oxidanylidene-pyrido[2,3-b][1,5]benzoxazepin-6-yl)ethanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |