| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLEC |
1-(4-amino-1,2,5-oxadiazol-3-yl)-5-[[cyclohexyl(methyl)amino]methyl]-N-[(4-fluorophenyl)methylideneamino]triazole-4-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(1-Benzyl-1H-pyrrolo[2,3-b]quinoxalin-2-yl)-4-chloro-benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-[4-(2-oxochromen-3-yl)-1,3-thiazol-2-yl]furan-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(1,3-benzodioxol-5-ylmethyl)-2-(3,4,5-trimethoxyphenyl)acetamide |
NA |
104814.2|200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
4-[3-(4-Methylphenoxy)propyl]morpholine |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-homoveratryl-4-keto-4-(6-methyl-2,3-dihydro-1,4-benzoxazin-4-yl)butyramide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-[(3-keto-4H-1,4-benzoxazin-6-yl)sulfonyl]-N-(2-methylcyclohexyl)propionamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
4-bromo-N-[(3-bromophenyl)methylideneamino]benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2,5-dichloro-N-[3-(4-morpholin-4-ylanilino)quinoxalin-2-yl]benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-[[4,5-Bis(dimethylamino)naphthalen-1-yl]methylidene]propanedinitrile |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-(4-bromo-8-chloronaphthalen-1-yl)sulfanyl-N-[4-(1,3-thiazol-2-ylsulfamoyl)phenyl]acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-[1-(2-fluorobenzyl)piperidin-3-yl]-3-(3-methoxyphenyl)-N-methylpropanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
(5-phenyl-1,3,4-oxadiazol-2-yl)methyl (E)-3-(furan-2-yl)prop-2-enoate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
4-[[[4-[(2,2-Dioxo-2lambda6-thia-3-azatricyclo[6.3.1.04,12]dodeca-1(11),4,6,8(12),9-pentaen-3-yl)methyl]benzoyl]hydrazinylidene]methyl]benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-chloro-N-[2-chloro-5-(trifluoromethyl)phenyl]-6-(3,5-dimethylpyrazol-1-yl)pyridine-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-[[3-chloro-5-(trifluoromethyl)pyridin-2-yl]sulfanylmethyl]-5-methyl-4-oxo-3H-thieno[2,3-d]pyrimidine-6-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
5-[(5E)-5-(3,4-dibenzoxybenzylidene)-4-keto-2-thioxo-thiazolidin-3-yl]valeric acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-[1-(4-imidazol-1-ylphenyl)ethyl]-2-methylsulfanylbenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-Quinolinecarbonitrile, 1,2-dihydro-1-benzoyl- |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-[4-[[5-(4-chlorophenyl)-6-ethoxycarbonyl-7-methyl-3-oxo-5H-thiazolo[3,2-a]pyrimidin-2-ylidene]methyl]phenoxy]acetic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |