| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLEC |
N-(2,5-dimethoxyphenyl)-N'-(4-methoxybenzyl)thiourea |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
1-[3-(Furan-2-ylmethylsulfanyl)-4-nitrophenyl]-4-methylsulfonylpiperazine |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-(2-Chlorophenyl)-6-[[4-(diethylamino)phenyl]methylidene]-[1,3]thiazolo[2,3-c][1,2,4]triazol-5-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(4-chlorobenzyl)-4,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-1-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(4-acetylphenyl)-2-(3-oxo-1,2,3,4-tetrahydronaphtho[1,8-ef][1,4]diazepin-2-yl)acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(2-morpholin-4-yl-5-nitrophenyl)thiophene-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-(3-oxo-1,2,3,4-tetrahydronaphtho[1,8-ef][1,4]diazepin-2-yl)-N-phenylacetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(4-chloro-2-methylphenyl)-2-[4-[hydroxy(diphenyl)methyl]piperidin-1-yl]acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
1,5-Dimethyl-4-[(4-oxocyclohexa-2,5-dien-1-ylidene)amino]-2-phenylpyrazol-3-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
4-(Benzylamino)naphthalene-1,2-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(2,4-dimethylphenyl)-4-[2-(2-nitrobenzoyl)hydrazinyl]-4-oxobutanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-[2-(benzylamino)-1-(4-methoxyphenyl)-2-oxoethyl]-N-(furan-2-ylmethyl)pyrazine-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
1-Benzhydryl-4-[(1-cyclopentyltetrazol-5-yl)-pyridin-2-ylmethyl]piperazine |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
4-[5-(3,4-Dimethoxyphenyl)triazol-1-yl]aniline |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-Benzenesulfonylamino-1-butyl-1H-pyrrolo[2,3-b]quinoxaline-3-carboxylic acid ethyl ester |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-[(2,4-Dichlorophenyl)sulfanyl]-1-(2,7-dimethylimidazo[1,2-a]pyridin-3-yl)-1-ethanone |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
1,2,2-Trimethyl-3-[(4-methyl-1-piperidinyl)carbonyl]cyclopentanecarboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
5-(3-chlorophenyl)-N-(2-piperidin-1-ylphenyl)furan-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(3-Benzenesulfonyl-1-butyl-1H-pyrrolo[2,3-b]quinoxalin-2-yl)-4-methyl-benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(2-adamantylideneamino)-4-methyl-3-nitrobenzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |