| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLEC |
N-[2-(3,4-dimethoxyphenyl)ethyl]-4-[methyl(phenyl)sulfamoyl]benzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-indol-1-yl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-[(1,2-dimethylindol-5-yl)methyl]-4-piperidin-1-ylsulfonylbenzamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
(5S)-5-[(3S,10R,13S)-3-hydroxy-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]-5-methyloxolan-2-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
(Z)-2-amino-3-[[4-(diethylamino)benzylidene]amino]but-2-enedinitrile |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
|
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
6-(piperidin-1-ylsulfonyl)-1,3-benzothiazol-2(3H)-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
1,1,3-Trimethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indol-2-ylidene)-propenyl]-1H-benzo[e]indolium |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-[[(E)-2-cyano-3-[3-ethoxy-4-(4-methylbenzoyl)oxyphenyl]prop-2-enoyl]amino]benzoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
4-[1-[(3-Methylphenyl)methoxy]-3-phenylpropan-2-yl]-1-(4-methylphenyl)sulfonyl-1,4-diazepan-5-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
Methyl 1-[4-[(2-chlorophenyl)methoxy]phenyl]-5-oxopyrrolidine-3-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
4-[(3-Chloro-1-benzothiophen-2-yl)methylideneamino]phenol |
NA |
127882.2 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
[4-[(E)-2-(1H-benzimidazol-2-yl)-2-cyanoethenyl]-2-methoxyphenyl] furan-2-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
(5Z)-3-butan-2-yl-5-[[9-methyl-4-oxo-2-(3-propan-2-yloxypropylamino)pyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-cyclohexyl-3-[(4-methylbenzoyl)amino]-9-azabicyclo[3.3.1]nonane-9-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-{(3,4-Dihydro-1H-isoquinolin-2-yl)-[1-(2-methoxy-ethyl)-1H-tetrazol-5-yl]-methyl}-7-methoxy-1H-quinolin-2-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-(4-benzylpiperazin-1-yl)-N-(3-chlorophenyl)propanamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
5-bromo-N-(3-cyano-1-phenyl-1H-pyrrolo[2,3-b]quinoxalin-2-yl)furan-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
1-(1,1,1,3,3,3-Hexafluoro-2-methylpropan-2-yl)-3-(4-hydroxyphenyl)urea |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
6-Ethylbenzo[b][1,4]benzothiazepine-3-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |