Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLG [5-[4-[(4-Carbamimidoylphenyl)methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(2-piperidin-4-ylethylcarbamoyl)piperazine-1-carboxylate 287000 NA NA NA NA NA BindingDB|TTD
PLG 2-Chloro-benzenesulfonic acid 3-methyl-5-[2-(methyl-pyridin-4-yl-amino)-ethoxy]-phenyl ester 200000 NA NA NA NA NA TTD
PLG 3-(6-chloronaphthalen-2-yl)sulfonyl-N-methyl-N-[1-(2-methylpyridin-4-yl)piperidin-4-yl]propanamide 200000 NA NA NA NA NA TTD
PLG 2-Acetylamino-N-[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-3-hydroxy-propionamide 1000000 NA NA NA NA NA TTD
PLG 2-methylpropyl 4-[[(2S)-2-[[4-(aminomethyl)cyclohexanecarbonyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]benzoate NA 370000 NA NA NA NA BindingDB
PLG H-Cys(1)-Pro-Ala-Tyr-Ser-Arg-Tyr-Leu-Asp-Cys(1)-OH 1000000 NA NA NA NA NA TTD
PLG N-(5-Methyl-pyridin-2-yl)-guanidine 245000 NA NA NA NA NA BindingDB|TTD
PLG N-[4-(6-Methylene-2-oxo-tetrahydro-pyran-3-yl)-benzyl]-guanidine 466000 NA NA NA NA NA BindingDB|TTD
PLG (1-{[(4-Carbamimidoyl-benzylcarbamoyl)-methyl]-carbamoyl}-2-hydroxy-ethyl)-carbamic acid tert-butyl ester 210000 NA NA NA NA NA BindingDB|TTD
PLG (4-{2-[(4-Aminomethyl-cyclohexanecarbonyl)-amino]-3-phenyl-propionylamino}-phenyl)-acetic acid NA 620000 NA NA NA NA BindingDB|TTD
PLG (S)-1-(3,3-Diphenyl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA 744000 NA NA NA NA NA BindingDB|TTD
PLG (2S)-N-cyclopentyl-N-methyl-5-[4-(methylamino)phenyl]-2-(5,6,7,8-tetrahydronaphthalen-2-ylsulfonylamino)pent-4-ynamide 200000 NA NA NA NA NA TTD
PLG 1-(2-Amino-3,3-dicyclohexyl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide 165000 NA NA NA NA NA BindingDB|TTD
PLG (2S)-N-cyclopentyl-N-methyl-5-[4-(methylamino)phenyl]-2-[(4-propylphenyl)sulfonylamino]pent-4-ynamide 200000 NA NA NA NA NA TTD
PLG (2S)-N-[(2S)-5-(diaminomethylideneamino)-1-oxopentan-2-yl]-1-(1,2,3,4-tetrahydroquinoline-2-carbonyl)pyrrolidine-2-carboxamide NA 660000 NA NA NA NA BindingDB|TTD
PLG 2-{(R)-3-[(R)-3-((S)-2-Benzyloxycarbonylamino-3-phenyl-propionylamino)-2-oxo-cyclohexyl]-propionylamino}-3-phenyl-propionic acid 3000000 NA NA NA NA NA BindingDB|TTD
PLG [5-[4-[(4-Carbamimidoylphenyl)methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(4-piperidin-4-ylbutanoyl)piperazine-1-carboxylate 310000 NA NA NA NA NA BindingDB|TTD
PLG (S)-1-((R)-2-Amino-2-cyclohexyl-acetyl)-pyrrolidine-2-carboxylic acid 5-chloro-2-cyclopropylcarbamoylmethoxy-benzylamide 113000 NA NA NA NA NA BindingDB|TTD
PLG 2-((R)-3-{(R)-3-[(S)-2-Benzyloxycarbonylamino-3-(1H-indol-3-yl)-propionylamino]-2-oxo-cyclohexyl}-propionylamino)-3-phenyl-propionic acid 150000 NA NA NA NA NA BindingDB
PLG 3-[Bis-(6-amino-hexyl)-amino]-tetrahydro-thiopyran-4-one 400000 NA NA NA NA NA BindingDB|TTD