| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLG |
(S)-1-(2-Amino-2-cyclohexyl-acetyl)-pyrrolidine-2-carboxylic acid 2,5-dichloro-benzylamide |
691000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
3-(4-Carbamimidoyl-phenyl)-2-[2-(4-cyano-benzenesulfonylamino)-acetylamino]-propionic acid ethyl ester |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
(S)-1-(2-5H-Dibenzo[a,d]cyclohepten-5-yl-acetyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; hydrochloride |
414000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
2-[2-(4-Carbamimidoyl-benzenesulfonylamino)-acetylamino]-3-(3-carbamimidoyl-phenyl)-propionic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
(S)-1-(3,3-Dicyclohexyl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; hydrochloride |
176000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
(S)-1-((R)-2-Amino-2-cyclohexyl-acetyl)-pyrrolidine-2-carboxylic acid 2-carbamoylmethoxy-5-chloro-benzylamide |
152000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
(S)-1-[(R)-2-Cyclohexyl-2-(diethylcarbamoylmethyl-amino)-acetyl]-pyrrolidine-2-carboxylic acid 2,5-dichloro-benzylamide |
244000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
3-(4-Carbamimidoyl-phenyl)-2-[2-(4-thiocarbamoyl-benzenesulfonylamino)-acetylamino]-propionic acid ethyl ester |
160000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
benzyl N-(4-amino-1-diphenoxyphosphorylbutyl)carbamate |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
2-Phenyl-1H-benzoimidazole-5-carboxamidine |
350000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
5-(4-Methyl-piperidin-4-yl)-isoxazol-3-ol; hydrobromide |
NA |
146000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
2-[[6-Amino-3-chloro-5-(diaminomethylidenecarbamoyl)pyrazin-2-yl]amino]acetic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
4-Nitrobenzamidine |
3981071.71 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
2-[4-[(3,3-dimethyl-2,4-dihydro-1H-quinolin-8-yl)sulfonylamino]-5-[4-(2-hydroxyethyl)piperidin-1-yl]-5-oxopentyl]guanidine |
210000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
Dehydroradiosumin |
NA |
209000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLG |
2-((R)-3-{(R)-3-[(S)-2-((S)-Benzyloxycarbonylamino)-3-phenyl-propionylamino]-2-oxo-cyclohexyl}-propionylamino)-3-(1H-indol-3-yl)-propionic acid |
420000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
N-Methyl-N-{3-[2-(pyridin-4-ylamino)-ethoxy]-phenyl}-benzenesulfonamide |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
N-[(2S)-3-(1,3-benzothiazol-2-yl)-1-[4-(2-hydroxyethyl)piperidin-1-yl]-1-oxopropan-2-yl]-3-methyl-1,2,3,4-tetrahydroquinoline-8-sulfonamide |
109000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
N-[(1S)-5-amino-1-cyanopentyl]-7-methyl-6-[[3-(3-methyl-2-oxo-1,3-benzoxazol-6-yl)-2,5-dioxoimidazolidin-1-yl]methyl]pyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-3-(2-oxo-3-propyl-1,3-benzoxazol-6-yl)imidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |