| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLEC |
N4-Sulfanilylsulfanilamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
5-(1-naphthylmethyl)-4-phenyl-4H-1,2,4-triazole-3-thiol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
|
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
1-(ethylamino)-3-methyl-3H-naphtho[1,2,3-de]quinoline-2,7-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
4-acetyl-N-[4-(3-methyl-[1,2,4]triazolo[4,3-b]pyridazin-6-yl)phenyl]benzenesulfonamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-(Azepan-1-ylmethylideneamino)-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridine-3-carbonitrile |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
|
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
4,6-Dimethyl-2-[(2-methylphenyl)amino]pyridine-3-carbonitrile |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-[2-(5-chloro-3-ethyl-1,3-benzothiazol-3-ium-2-yl)ethenyl]-N-methylaniline |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
|
NA |
100420|200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
(E)-3-(2-chloro-6-fluorophenyl)-2-cyano-N-cyclopropylprop-2-enamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(4-chlorobenzyl)-N-[3-(methylsulfanyl)-1H-1,2,4-triazol-5-yl]amine |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-Amino-4-(ethylamino)benzoic acid |
NA |
133137.4 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
methyl 5-benzamido-6-oxidanylidene-2-[(E)-2-[(4-phenoxyphenyl)amino]ethenyl]pyran-3-carboxylate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
2-hydroximino-N-[2-(1-methylpiperidin-1-ium-1-yl)ethyl]acetamide;iodide |
NA |
129726.9|200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
4-(4-Hydroxyanilino)-1-(4-hydroxyphenyl)-2-methyl-5-oxo-2-pyrrolecarboxylic acid ethyl ester |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
8-(4-ET-1-Piperazinyl)-3-ME-7-(2-ME-2-propenyl)-3,7-dihydro-1H-purine-2,6-dione |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
N-(2-chlorobenzyl)-4-keto-1-methyl-6-(4-methylpiperidino)sulfonyl-quinoline-3-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
1-[(3,4-Difluorobenzylidene)amino]-3-(3-pyridyl)thiourea |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLEC |
3-(2,3-dihydro-1H-indol-1-ylcarbonyl)-8-methoxy-2H-chromen-2-one |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |