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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLG 2-[[6-amino-3-chloro-5-[(Z)-N'-hydroxycarbamimidoyl]pyrazin-2-yl]amino]acetic acid NA 250000 NA NA NA NA TTD
PLG 2-(3,4-Dihydroxyphenyl)-5-[[4-[[2-(3,4-dihydroxyphenyl)-3,7-dihydroxy-4-oxochromen-5-yl]oxymethyl]phenyl]methoxy]-3,7-dihydroxychromen-4-one NA 116000 NA NA NA NA BindingDB|TTD
PLG tetrasodium;[4-[4-oxo-5-[(E)-4-[4-oxo-7-sulfonatooxy-2-(4-sulfonatooxyphenyl)chromen-5-yl]oxybut-2-enoxy]-7-sulfonatooxychromen-2-yl]phenyl] sulfate NA 121000 NA NA NA NA BindingDB|TTD
PLG Tetrasodium;[4-[4-oxo-5-[4-[4-oxo-7-sulfonatooxy-2-(4-sulfonatooxyphenyl)chromen-5-yl]oxybutoxy]-7-sulfonatooxychromen-2-yl]phenyl] sulfate NA 282000 NA NA NA NA BindingDB|TTD
PLG Tetrasodium;[4-[4-oxo-5-[3-[4-oxo-7-sulfonatooxy-2-(4-sulfonatooxyphenyl)chromen-5-yl]oxypropoxy]-7-sulfonatooxychromen-2-yl]phenyl] sulfate NA 1000000 NA NA NA NA TTD
PLG Octasodium;[2-(3,4-disulfonatooxyphenyl)-5-[[6-[[2-(3,4-disulfonatooxyphenyl)-4-oxo-3,7-disulfonatooxychromen-5-yl]oxymethyl]pyridin-2-yl]methoxy]-4-oxo-3-sulfonatooxychromen-7-yl] sulfate NA 231000 NA NA NA NA BindingDB|TTD
PLG (2S)-6-amino-2-[(4-methylphenyl)sulfonylamino]-N-(4-nitrophenyl)hexanamide NA 700000 NA NA NA NA BindingDB|TTD
PLG Xeruborbactam NA 1000000 NA NA NA NA PubChem
PLG benzyl N-[(5S)-5-[[4-(aminomethyl)cyclohexanecarbonyl]amino]-7-(4-benzoylphenoxy)-6-oxoheptyl]carbamate NA 200000 NA NA NA NA BindingDB|TTD
PLG Naphthalene-2-sulfonic acid {3-[2-(pyridin-4-ylamino)-ethoxy]-phenyl}-amide 500000 NA NA NA NA NA TTD
PLG 4-Chloro-N-{3-[2-(pyridin-4-ylamino)-ethoxy]-phenyl}-benzenesulfonamide 500000 NA NA NA NA NA TTD
PLG 4-[2-(3-Benzenesulfonylamino-phenoxy)-ethylamino]-pyridinium 500000 NA NA NA NA NA TTD
PLG N-[(2S)-6-amino-1-[(4-benzoylphenoxy)methylamino]-1-oxohexan-2-yl]-4-(aminomethyl)cyclohexane-1-carboxamide NA 660000 NA NA NA NA BindingDB|TTD
PLG (2S)-6-amino-N-(4-benzoylphenyl)-2-[(4-methylphenyl)sulfonylamino]hexanamide NA 140000 NA NA NA NA BindingDB|TTD
PLG Phenylguanidine 2610000 NA NA NA NA NA BindingDB|TTD
PLG Benzamidine HCl hydrate 501187.23 NA NA NA NA NA TTD
PLG Amiloride NA 250000 NA NA NA NA PubChem
PLG 4-(2-Aminoethyl)benzenesulfonylfluoride NA 240000 NA NA NA NA BindingDB|TTD
PLG Dalfampridine 2000000 NA NA NA NA NA PubChem|TTD
PLG 4-(2-Hydroxyethylamino)-pyridine 500000 NA NA NA NA NA TTD