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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLG 130000 NA NA NA NA NA BindingDB
PLG [Amino({4-[(3-hydroxynaphthalene-2-)amido]phenyl}amino)methylidene]azanium 130000 NA NA NA NA NA BindingDB
PLG Diphenyl 1-(2,3,6-tri-isopropylbenzenesulfonyl)amino-2-(4-guanidinophenyl)-ethanephosphonate NA 125000 NA NA NA NA BindingDB|TTD
PLG 1-Ethyl-1H-indole-5-carboxamidine 400000 NA NA NA NA NA TTD
PLG 1-Benzyl-1H-indole-5-carboxamidine 844000 NA NA NA NA NA BindingDB|TTD
PLG 3-Amidinophenylpyruvic acid 2510000|1584893.19 NA NA NA NA NA BindingDB|TTD
PLG 3,5-Dimethylbenzenecarboximidamide 250000|251188.64 NA NA NA NA NA BindingDB|TTD
PLG 3-Phenylbenzenecarboximidamide 3160000|316227.77 NA NA NA NA NA BindingDB|TTD
PLG LY 806303 NA 240000 NA NA NA NA BindingDB|TTD
PLG 3-(Aminoiminomethyl)benzoic acid 1580000|398107.17 NA NA NA NA NA BindingDB|TTD
PLG 3-(Hydroxymethyl)benzene-1-carboximidamide 398000|2511886.43 NA NA NA NA NA BindingDB|TTD
PLG (2S)-N-cyclopentyl-N-methyl-5-[4-(methylamino)phenyl]-2-(naphthalen-2-ylsulfonylamino)pent-4-ynamide 200000 NA NA NA NA NA TTD
PLG (2S)-N-cyclopentyl-2-[(6-methoxynaphthalen-2-yl)sulfonylamino]-N-methyl-5-[4-(methylamino)phenyl]pent-4-ynamide 200000 NA NA NA NA NA TTD
PLG N-[3-(1,3-benzothiazol-2-yl)-1-(4-ethylpiperidin-1-yl)-1-oxopropan-2-yl]-3,3-dimethyl-2,4-dihydro-1H-quinoline-8-sulfonamide 240000 NA NA NA NA NA BindingDB|TTD
PLG 2-Chloro-benzenesulfonic acid 3-(5-guanidino-pentyloxy)-5-methyl-phenyl ester 200000 NA NA NA NA NA TTD
PLG 2-Chloro-benzenesulfonic acid 3-(1-carbamimidoyl-piperidin-3-ylmethoxy)-5-methyl-phenyl ester 200000 NA NA NA NA NA TTD
PLG 2-Chloro-benzenesulfonic acid 3-(3-guanidino-propoxy)-5-methyl-phenyl ester 200000 NA NA NA NA NA TTD
PLG 2-Chloro-benzenesulfonic acid 3-(4-guanidino-butoxy)-5-methyl-phenyl ester 200000 NA NA NA NA NA TTD
PLG {[2-(1-Carbamimidoyl-piperidin-4-yl)-ethylcarbamoyl]-methyl}-carbamic acid 4-{[2-(1-carbamimidoyl-piperidin-4-yl)-ethylcarbamoyl]-methylcarbamoyloxymethyl}-benzyl ester 1000000 NA NA NA NA NA TTD
PLG {[(1-Carbamimidoyl-piperidin-4-ylmethyl)-carbamoyl]-methyl}-carbamic acid 4-{[(1-carbamimidoyl-piperidin-4-ylmethyl)-carbamoyl]-methylcarbamoyloxymethyl}-benzyl ester 1000000 NA NA NA NA NA TTD