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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLG [5-[4-[[4-[(E)-N'-methoxycarbonylcarbamimidoyl]phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(2-piperidin-4-ylethylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG 1,4-Di[4-(4-aminomethylhexahydro-1-pyridinylcarboxamidomethyl)hexahydro-1-pyridinylcarbonyloxymethyl]benzene 1000000 NA NA NA NA NA TTD
PLG {4-[(4-Aminomethyl-piperidine-1-carbonyl)-amino]-butyl}-carbamic acid 4-{4-[(4-aminomethyl-piperidine-1-carbonyl)-amino]-butylcarbamoyloxymethyl}-benzyl ester 1000000 NA NA NA NA NA TTD
PLG [5-[4-(2-Piperidin-4-ylethylcarbamoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-[2-(4-carbamimidoylphenyl)acetyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[2-(4-Carbamimidoylanilino)-2-oxoethyl]piperidine-1-carbonyl]oxycyclooctyl] 4-(2-piperidin-4-ylethylcarbamoyl)piperazine-1-carboxylate 293000 NA NA NA NA NA BindingDB|TTD
PLG [5-[4-[[(4-Carbamimidoylphenyl)sulfonylamino]methyl]piperidine-1-carbonyl]oxycyclooctyl] 4-(2-piperidin-4-ylethylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[(4-Carbamimidoylbenzoyl)amino]methyl]piperidine-1-carbonyl]oxycyclooctyl] 4-(2-piperidin-4-ylethylcarbamoyl)piperazine-1-carboxylate 279000 NA NA NA NA NA BindingDB|TTD
PLG [5-[4-[[(4-Carbamimidoylbenzoyl)amino]methyl]piperidine-1-carbonyl]oxycyclooctyl] 4-(4-piperidin-4-ylbutanoyl)piperazine-1-carboxylate 320000 NA NA NA NA NA BindingDB|TTD
PLG (E)-3-(5-Chloro-2-guanidino-pyridin-3-yl)-acrylic acid 278500 NA NA NA NA NA BindingDB|TTD
PLG N-(5-Chloro-3-phenylethynyl-pyridin-2-yl)-guanidine 218000 NA NA NA NA NA BindingDB|TTD
PLG 3-Hydroxy-anthracene-2-carboxylic acid (4-guanidino-phenyl)-amide 283000 NA NA NA NA NA BindingDB|TTD
PLG 3-Bromo-N-(4-guanidino-phenyl)-2-hydroxy-5-methyl-benzamide 205000 NA NA NA NA NA BindingDB|TTD
PLG [5-[4-[[4-(Aminomethyl)-1-bicyclo[2.2.2]octanyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[[4-(aminomethyl)-1-bicyclo[2.2.2]octanyl]methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[(4-aminocyclohexyl)methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [3-[[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxymethyl]-1-adamantyl]methyl 4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carboxylate 576000 NA NA NA NA NA BindingDB|TTD
PLG [5-[4-[2-(4-Carbamimidoylphenyl)acetyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-(4-carbamimidoylphenyl)acetyl]piperazine-1-carboxylate 155000 NA NA NA NA NA BindingDB|TTD
PLG [5-[4-(6-Imidazol-1-ylhexanoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(6-imidazol-1-ylhexanoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-(4-Piperidin-4-ylbutanoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(4-piperidin-4-ylbutanoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG N-[[4-(aminomethyl)phenyl]methyl]-N'-[[4-[[[4-[[4-(aminomethyl)phenyl]methylamino]-4-oxobutanoyl]amino]methyl]phenyl]methyl]butanediamide 769000 NA NA NA NA NA BindingDB|TTD
PLG N-[[4-(aminomethyl)phenyl]methyl]-N'-[[4-[[[4-[[4-(aminomethyl)phenyl]methylamino]-4-oxobutanoyl]-methylamino]methyl]phenyl]methyl]-N'-methylbutanediamide 214000 NA NA NA NA NA BindingDB|TTD