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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLG N'-[[4-(aminomethyl)phenyl]methyl]-N-[[4-[[[4-[[4-(aminomethyl)phenyl]methyl-methylamino]-4-oxobutanoyl]amino]methyl]phenyl]methyl]-N'-methylbutanediamide 1000000 NA NA NA NA NA TTD
PLG N'-[[4-(diaminomethylideneamino)phenyl]methyl]-N-[[4-[[[3-[[4-(diaminomethylideneamino)phenyl]methylamino]-3-oxopropanoyl]amino]methyl]phenyl]methyl]propanediamide 1000000 NA NA NA NA NA TTD
PLG [5-[4-[2-(1-Ethanimidoylpiperidin-4-yl)ethylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-(1-ethanimidoylpiperidin-4-yl)ethylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[(1-Ethanimidoylpiperidin-4-yl)methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[(1-ethanimidoylpiperidin-4-yl)methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG N-[[4-(aminomethyl)phenyl]methyl]-N'-[[4-[[[3-[[4-(aminomethyl)phenyl]methylamino]-3-oxopropanoyl]amino]methyl]phenyl]methyl]propanediamide 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(3-piperidin-4-ylpropylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(2-piperidin-4-ylethylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(piperidin-4-ylmethylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Aminomethyl)cyclohexyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[[4-(aminomethyl)cyclohexyl]methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [(2S,3S)-3-[[4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxymethyl]-2-bicyclo[2.2.2]oct-5-enyl]methyl 4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carboxylate 700000 NA NA NA NA NA BindingDB|TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(4-piperidin-4-ylbutanoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(2-pyridin-4-ylethylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [4-[[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxymethyl]phenyl]methyl 4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxy-1,2,3,3a,4,5,6,6a-octahydropentalen-2-yl] 4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG Pentanedioic acid 4-guanidino-benzylamide 4-{[4-(4-guanidino-benzylcarbamoyl)-butyrylamino]-methyl}-benzylamide 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(benzylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[2-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoylamino]acetyl]oxycyclooctyl] 2-[[4-(diaminomethylideneamino)phenyl]methylcarbamoylamino]acetate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-(1-methylpiperidin-4-yl)ethylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[Methyl(2-piperidin-4-ylethyl)carbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG N-[[4-(diaminomethylideneamino)phenyl]methyl]-4-[10-[4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazin-1-yl]-10-oxodecanoyl]piperazine-1-carboxamide 1000000 NA NA NA NA NA TTD