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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(5-imidazol-1-ylpentanoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG (1R,6S,8S,8aS)-6-Amino-6-cyclohex-1-enylmethyl-1-ethyl-8-methoxy-5-oxo-octahydro-indolizine-3-carboxylic acid 4-carbamimidoyl-benzylamide; hydrochloride NA 141000 NA NA NA NA BindingDB|TTD
PLG 1-(4-Carbamimidoyl-2-chloro-benzyl)-1H-indole-5-carboxamidine 700000 NA NA NA NA NA TTD
PLG 3-Benzoyl-1H-indole-6-carboxamidine 200000 NA NA NA NA NA TTD
PLG 4-(5-Nitro-indol-1-ylmethyl)-benzamidine 400000 NA NA NA NA NA TTD
PLG 3-(2,2,2-Trifluoro-acetyl)-1H-indole-6-carboxamidine 1000000 NA NA NA NA NA TTD
PLG 3-Acetyl-1H-indole-6-carboxamidine 1000000 NA NA NA NA NA TTD
PLG 1-(3-Amino-benzyl)-1H-indole-5-carboxamidine 164000 NA NA NA NA NA BindingDB|TTD
PLG (2R)-2-amino-N-[(2S)-1-[6-aminohexyl(cyclohexyl)amino]-1-oxo-3-phenylpropan-2-yl]-3-methylpentanamide 520000 NA NA NA NA NA BindingDB|TTD
PLG {2-[2-(1-Formyl-4-guanidino-butylcarbamoyl)-pyrrolidin-1-yl]-1-phenyl-ethyl}-carbamic acid tert-butyl ester NA 400000 NA NA NA NA BindingDB|TTD
PLG (2S)-N-[5-(diaminomethylideneamino)-1-oxopentan-2-yl]-1-(1H-indole-2-carbonyl)pyrrolidine-2-carboxamide NA 420000 NA NA NA NA BindingDB
PLG (2S)-N-[5-(diaminomethylideneamino)-1-oxopentan-2-yl]-1-[(2S)-2-methoxy-2-phenylacetyl]pyrrolidine-2-carboxamide NA 860000 NA NA NA NA BindingDB
PLG N-(5-Bromo-isoquinolin-1-yl)-guanidine 237800 NA NA NA NA NA BindingDB|TTD
PLG N-(6-Bromo-isoquinolin-1-yl)-guanidine 131400 NA NA NA NA NA BindingDB|TTD
PLG (S)-1-(3-Phenyl-3-pyridin-4-yl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA 744000 NA NA NA NA NA BindingDB|TTD
PLG (S)-1-(3-Phenyl-3-pyridin-3-yl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA 1000000 NA NA NA NA NA TTD
PLG (S)-1-(3-Phenyl-3-pyridin-2-yl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA 1000000 NA NA NA NA NA TTD
PLG (S)-1-(3-Benzo[1,3]dioxol-5-yl-3-pyridin-3-yl-propionyl)-pyrrolidine-2-carboxylic acid (4-amino-cyclohexylmethyl)-amide; TFA 572000 NA NA NA NA NA BindingDB|TTD
PLG H-Tic-Pro-aMeArg-al NA 740000 NA NA NA NA BindingDB|TTD
PLG Me-Phe-Pro-aMeArg-al NA 850000 NA NA NA NA BindingDB|TTD