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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLG N-[(4-Carbamimidoyl-benzylcarbamoyl)-methyl]-3-hydroxy-2-(2-phenyl-ethenesulfonylamino)-propionamide 140000 NA NA NA NA NA BindingDB|TTD
PLG 4-tert-Butoxycarbonylamino-4-{[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-carbamoyl}-butyric acid 1000000 NA NA NA NA NA TTD
PLG Boc-D-Ser-Gly-NHBn(4-amidino) 1000000 NA NA NA NA NA TTD
PLG 3-Hydroxy-N-{[4-(N-hydroxycarbamimidoyl)-benzylcarbamoyl]-methyl}-2-phenylmethanesulfonylamino-propionamide 1000000 NA NA NA NA NA TTD
PLG (1-{[(4-Carbamimidoyl-benzylcarbamoyl)-methyl]-carbamoyl}-2-hydroxy-ethyl)-carbamic acid benzyl ester 160000 NA NA NA NA NA BindingDB|TTD
PLG (4-Guanidino-benzyl)-carbamic acid benzyl ester 1000000 NA NA NA NA NA TTD
PLG 2-(4-Chloro-benzenesulfonylamino)-N-[(R)-1-(piperidine-1-carbonyl)-3-(pyridin-4-ylamino)-propyl]-acetamide 500000 NA NA NA NA NA TTD
PLG 2-Benzenesulfonylamino-N-[(R)-1-(piperidine-1-carbonyl)-3-(pyridin-4-ylamino)-propyl]-acetamide 500000 NA NA NA NA NA TTD
PLG N-(2-phenoxyethyl)pyridin-4-amine 500000 NA NA NA NA NA TTD
PLG 2-(Naphthalene-2-sulfonylamino)-N-[(R)-1-(piperidine-1-carbonyl)-3-(pyridin-4-ylamino)-propyl]-acetamide 500000 NA NA NA NA NA TTD
PLG 2-(Naphthalene-2-sulfonylamino)-N-[(S)-1-(piperidine-1-carbonyl)-3-(pyridin-4-ylamino)-propyl]-acetamide 500000 NA NA NA NA NA TTD
PLG Pyridin-4-yl-(2-m-tolyloxy-ethyl)-amine 500000 NA NA NA NA NA TTD
PLG 4-(Hydroxymethyl)Benzamidine 9990000|630957.34 NA NA NA NA NA BindingDB|TTD
PLG (S)-N-((1-carbamimidoylpiperidin-4-yl)methyl)-5-guanidino-2-((S)-2-((S)-5-guanidino-2-(2-phenylacetamido)pentanamido)-3-methylbutanamido)pentanamide 1000000 NA NA NA NA NA TTD
PLG 3-Bromo-benzamidine 7943282.35 NA NA NA NA NA TTD
PLG 5-[(2R,4R)-2-benzylpiperidin-4-yl]-1,2-oxazol-3-one NA 169000 NA NA NA NA BindingDB|TTD
PLG 5-[(2S,4R)-2-benzylpiperidin-4-yl]-1,2-oxazol-3-one NA 150000 NA NA NA NA BindingDB|TTD
PLG 3-[2-Amino-3-(4-methanesulfonyl-piperazin-1-yl)-3-oxo-propyl]-benzamidine 1000000 NA NA NA NA NA TTD
PLG 3-Methoxy-benzamidine 630000|1580000|316227.77 NA NA NA NA NA BindingDB|TTD
PLG 3,4-Dimethylbenzene-1-carboximidamide 4000000|3162277.66 NA NA NA NA NA BindingDB|TTD