| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLG |
2-Methyl-benzamidine |
199000|316227.77 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
[Amino-(4-nitrophenyl)methylidene]azanium |
99900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLG |
2-[(6-Amino-5-carbamimidoylpyrazin-2-yl)amino]acetic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
Benzyl 2-[(6-amino-5-carbamoyl-3-chloropyrazin-2-yl)amino]acetate |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
2-[(6-Amino-5-carbamimidoyl-3-chloropyrazin-2-yl)amino]acetic acid |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
2-[[6-Amino-5-(diaminomethylidenecarbamoyl)pyrazin-2-yl]amino]acetic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
2-[[(1R,7S,13S,16S,19S,22R,34R,43S,49S)-34-[(2-aminoacetyl)amino]-43-[3-(diaminomethylideneamino)propyl]-19-[(4-hydroxyphenyl)methyl]-16-methyl-2,8,14,17,20,35,38,41,44,50-decaoxo-24,32,53-trithia-3,9,15,18,21,36,39,42,45,51-decazahexacyclo[26.23.3.126,30.03,7.09,13.045,49]pentapentaconta-26,28,30(55)-triene-22-carbonyl]amino]acetic acid |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
H-Ala-Cys-Asp-Ala-Arg-Pro-Cys-Pro-Gln-Thr-Tyr-Cys-Leu-OH |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
H-Gly-Cys-Leu-Gly-Arg-Pro-Cys-Pro-Met-Ala-Tyr-Cys-Ser-OH |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
H-Gln-Cys-Asn-Ala-Arg-Pro-Cys-Pro-Ser-Ser-Tyr-Cys-Arg-OH |
118300 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
H-Gly-Cys-Ala-Ala-Arg-Pro-Cys-Pro-Leu-Thr-Ala-Cys-Trp-OH |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
H-Gly-Cys-Trp-Ala-Arg-Pro-Cys-Pro-Leu-Ala-Leu-Cys-Gln-OH |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
H-Gly-Cys-Met-Gly-Arg-Pro-Cys-Pro-Val-Ser-Tyr-Cys-Phe-OH |
120000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
4-Amino-4-{[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-carbamoyl}-butyric acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
(R)-2-Amino-3-methyl-pentanoic acid [(S)-1-(4-oxo-tetrahydro-thiopyran-3-ylcarbamoyl)-2-phenyl-ethyl]-amide |
16000000|9000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
(2R,3S)-2-amino-N-[(2S)-1-[6-aminohexyl-(4-oxothian-3-yl)amino]-1-oxo-3-phenylpropan-2-yl]-3-methylpentanamide |
630000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLG |
N-[(1S)-5-amino-1-cyanopentyl]-7-methyl-6-[(3-methyl-2,5-dioxoimidazolidin-1-yl)methyl]pyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-(4-fluorophenyl)-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLG |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[3-(4-methoxyphenyl)-2,5-dioxoimidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
180000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-3-(4-propylphenyl)imidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
330000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |