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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLG (2R)-2-amino-N-[3,5-bis[(E)-N-(diaminomethylideneamino)-C-methylcarbonimidoyl]phenyl]-5-(diaminomethylideneamino)pentanamide 1000000 NA NA NA NA NA BindingDB|TTD
PLG N-(3,5-bis(-1-(2-carbamimidoylhydrazono)ethyl)phenyl)-4-guanidinobutanamide 1000000 NA NA NA NA NA BindingDB|TTD
PLG 2-[(E)-1-[3-(benzenesulfonamido)-5-[(E)-N-(diaminomethylideneamino)-C-methylcarbonimidoyl]phenyl]ethylideneamino]guanidine 400000 NA NA NA NA NA BindingDB|TTD
PLG N-(3,5-bis(-1-(2-carbamimidoylhydrazono)ethyl)phenyl)-5-guanidinopentanamide 1000000 NA NA NA NA NA BindingDB|TTD
PLG N-(3,5-bis(-1-(2-carbamimidoylhydrazono)ethyl)phenyl)-6-guanidinohexanamide 1000000 NA NA NA NA NA BindingDB|TTD
PLG amino-N-(3,5-bis(-1-(2-carbamimidoylhydrazono)ethyl)phenyl)butanamide 110000 NA NA NA NA NA BindingDB|TTD
PLG Tranexamic acid NA|25000000|40000000 NA|2000000|10000000|241000 750000|NA NA NA NA BindingDB|GtoPDB|PubChem
PLG Aminocaproic Acid NA|53000000 105000|NA NA NA NA NA BindingDB|PubChem|TTD
PLG Vaborbactam NA 1000000 NA NA NA NA PubChem|TTD
PLG H-D-Ile-Phe-Lys-NH2 NA 290000 NA NA NA NA BindingDB|TTD
PLG tert-butyl 3-[3-[5-[[(1S)-5-amino-1-cyanopentyl]carbamoyl]-2-(pyridin-4-ylmethoxy)anilino]-3-oxopropyl]indole-1-carboxylate NA 220000 NA NA NA NA BindingDB|TTD
PLG Methyl 3-[4-[(6-carbamoylnaphthalene-2-carbonyl)amino]phenyl]benzoate NA 125000 NA NA NA NA TTD
PLG N-[(1S)-5-amino-1-cyanopentyl]-3-[3-[1-[(4-fluorophenyl)methyl]indol-3-yl]propanoylamino]-4-(pyridin-4-ylmethoxy)benzamide NA 140000 NA NA NA NA BindingDB|TTD
PLG N-[(1S)-5-amino-1-cyanopentyl]-3-[(2-naphthalen-2-ylacetyl)amino]-4-(pyridin-4-ylmethoxy)benzamide NA 220000 NA NA NA NA BindingDB|TTD
PLG N-[(1S)-5-amino-1-cyanopentyl]-3-[3-(1H-indol-3-yl)propanoylamino]-4-(pyridin-4-ylmethoxy)benzamide NA 370000 NA NA NA NA BindingDB|TTD
PLG N-[(1S)-5-amino-1-cyanopentyl]-3-[[2-(4-fluorophenyl)acetyl]amino]-4-(pyridin-4-ylmethoxy)benzamide NA 590000 NA NA NA NA BindingDB|TTD
PLG N-[(1S)-5-amino-1-cyanopentyl]-3-[(2-naphthalen-1-ylacetyl)amino]-4-(pyridin-4-ylmethoxy)benzamide NA 570000 NA NA NA NA BindingDB|TTD
PLG N-[(1S)-5-amino-1-cyanopentyl]-4-(pyridin-4-ylmethoxy)benzamide NA 240000 NA NA NA NA BindingDB|TTD
PLG Benzyl 2-[(6-amino-5-carbamimidoyl-3-chloropyrazin-2-yl)amino]acetate NA 250000 NA NA NA NA TTD
PLG Benzyl 2-[[6-amino-3-chloro-5-(diaminomethylidenecarbamoyl)pyrazin-2-yl]amino]acetate NA 250000 NA NA NA NA TTD