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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLG (2S)-N-[(1R,2S)-3-cyclohexyl-1-hydroxy-1-(1,3-thiazol-2-yl)propan-2-yl]-2-[[(2S)-2-[4-(diaminomethylideneamino)butanoylamino]-3-phenylpropanoyl]amino]-4-methylpentanamide NA 143000 NA NA NA NA BindingDB|TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carboxylate 494000 NA NA NA NA NA BindingDB|TTD
PLG (3aalpha,6aalpha)-3beta,6beta-Bis[4-(4-guanidinobenzylcarbamoyl)piperazinocarbonyloxy]hexahydrofuro[3,2-b]furan 700000 NA NA NA NA NA BindingDB|TTD
PLG 2-Chloro-benzenesulfonic acid 3-(1-carbamimidoyl-piperidin-4-ylmethoxy)-5-methyl-phenyl ester 200000 NA NA NA NA NA TTD
PLG GW-813893 NA 158000 NA NA NA NA PubChem|TTD
PLG (2S)-2-amino-N-[2-[(4-carbamimidoylphenyl)methylamino]-2-oxoethyl]-3-hydroxypropanamide 1000000 NA NA NA NA NA TTD
PLG 2-Amino-N-[(4-carbamimidoyl-benzylcarbamoyl)-methyl]-3-hydroxy-propionamide 1000000 NA NA NA NA NA TTD
PLG CGH-1484A free base 212000 NA NA NA NA NA BindingDB|TTD
PLK1 (+/-)-Trachyspic acid NA 128000 NA NA NA NA BindingDB
PLK1 N,5-dimethyl-2-(3-morpholin-4-ylpropyl)-1-phenyl-2H-pyrrol-1-ium-4-carboxamide NA 550000 NA NA NA NA BindingDB|ChEMBL
PLK1 N-methyl-4-phenyl-5-(trifluoromethyl)thiophene-2-carboxamide NA 500000|5e+05 NA NA NA NA BindingDB|ChEMBL
PLK1 Trachyspic acid 19-butyl ester NA 102000 NA NA NA NA BindingDB
PLK1 1-(benzenesulfonyl)-N-methylindole-3-carboxamide NA 375000 NA NA NA NA BindingDB|ChEMBL
PLK1 3,6-dichloro-N-[(E)-(5-ethylthiophen-2-yl)methylideneamino]-1H-indene-2-carboxamide NA NA 251000 NA NA NA BindingDB
PLK1 3-carbazol-9-yl-N-[(E)-(3,5-dichlorophenyl)methylideneamino]propanamide NA NA 339000 NA NA NA BindingDB
PLK1 2-[2-(4-Octylphenyl)ethylamino]benzoic acid NA 117500 NA NA NA NA BindingDB
PLK1 4-octyl-N-(2-sulfamoylphenyl)benzamide NA 259100 NA NA NA NA BindingDB
PLK1 N-Methyl-1-naphthalenecarboxamide NA 104000 NA NA NA NA BindingDB|ChEMBL
PLK1 3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide NA 380000 NA NA NA NA ChEMBL
PLK1 4-methoxy-N-methylbenzamide NA 125000 NA NA NA NA BindingDB|ChEMBL