| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLK1 |
9-Chloro-2-[2-chloro-5-[3-(dimethylamino)propyl]anilino]-5,7-dihydropyrimido[5,4-d][1]benzazepine-6-thione |
NA |
NA |
NA |
440000 |
NA |
NA |
TTD |
| PLK1 |
9-Chloro-2-[3-chloro-5-[3-(dimethylamino)propyl]anilino]-5,7-dihydropyrimido[5,4-d][1]benzazepine-6-thione |
NA |
NA |
NA |
150000 |
NA |
NA |
TTD |
| PLK1 |
[(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(1-acetylpyrrolidine-2-carbonyl)amino]-4-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-2-methyl-4-oxobutyl]phosphonic acid |
NA |
174000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLK1 |
[(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(1-acetylpyrrolidine-2-carbonyl)amino]-4-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] 5-phenylpentyl hydrogen phosphate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLK1 |
[(2R,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[(1-acetylpyrrolidine-2-carbonyl)amino]-4-methylpentanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-hydroxypropanoyl]amino]-4-amino-4-oxobutan-2-yl] 9-phenylnonyl hydrogen phosphate |
NA |
154000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLK1 |
N-methylquinoline-6-carboxamide |
NA |
400000|4e+05 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PLK1 |
N-methyl-2-(6-methylthieno[2,3-d]pyrimidin-4-yl)sulfanylacetamide |
NA |
475000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PLK1 |
N,2-dimethyl-1,5-diphenylpyrrole-3-carboxamide |
NA |
600000|6e+05 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PLK1 |
N-methyl-2-[5-(4-methylphenyl)-2-oxopyrazin-1-yl]acetamide |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PLK1 |
N-[(E)-2,3-dihydro-1,4-benzodioxin-6-ylmethylideneamino]-2-(2-methylphenoxy)acetamide |
NA |
NA |
412000 |
NA |
NA |
NA |
BindingDB |
| PLK1 |
N'-(4-chlorobenzylidene)-2-[(2,6-dimethyl-4-quinolinyl)sulfanyl]acetohydrazide |
NA |
NA |
418000 |
NA |
NA |
NA |
BindingDB |
| PLK1 |
4-[2-(2-hydroxyethoxy)-5-methyl-3-[4-(2H-tetrazol-5-yl)phenyl]phenyl]benzonitrile |
NA |
139000|146000|151000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLK1 |
5-(3-methoxyphenyl)-N-methylpyrazolidine-3-carboxamide |
NA |
380000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLK1 |
2-[(4-Pentylbenzoyl)amino]benzoic acid |
NA |
223600 |
NA |
NA |
NA |
NA |
BindingDB |
| PLK1 |
Poloxin |
NA |
NA |
408000 |
NA |
NA |
NA |
BindingDB |
| PLK2 |
(2S)-dihydrobaicalein |
NA |
242200 |
NA |
NA |
NA |
NA |
BindingDB |
| PLK2 |
3-carbazol-9-yl-N-[(E)-(3,5-dichlorophenyl)methylideneamino]propanamide |
NA |
NA |
210000 |
NA |
NA |
NA |
BindingDB |
| PLK2 |
3-[[(1R,9S)-1,9-dimethyl-3-naphthalen-2-yl-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methyl]benzonitrile |
NA |
95500000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLK2 |
5-Hydroxy-7,8-dimethoxyflavone |
NA |
951900 |
NA |
NA |
NA |
NA |
BindingDB |
| PLK2 |
Baicalein |
NA |
314000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |