| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLK2 |
1-[(Z)-N-(benzenesulfonylmethyl)-C-(4-methylphenyl)carbonimidoyl]-3-(4-nitrophenyl)thiourea |
NA |
NA |
159000 |
NA |
NA |
NA |
BindingDB |
| PLK2 |
N-[(E)-2,3-dihydro-1,4-benzodioxin-6-ylmethylideneamino]-2-(2-methylphenoxy)acetamide |
NA |
NA |
197000 |
NA |
NA |
NA |
BindingDB |
| PLK3 |
(2S)-dihydrobaicalein |
NA |
1604000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLK3 |
5-Hydroxy-7,8-dimethoxyflavone |
NA |
5123000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLK3 |
Poloxin |
NA |
NA |
296000 |
NA |
NA |
NA |
BindingDB |
| PLTP |
N-(5-butyl-4-(4-methoxyphenyl)-1,3-selenazol-2-yl)-3,4,5-trimethoxybenzamide |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNLIP |
Koenigicine |
NA |
428600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNLIP |
methyl (2R)-2-[[(2E,8E)-deca-2,8-dienoyl]amino]-3-[(5R)-5-hydroxy-6-oxo-3,8-dioxatricyclo[5.1.0.02,4]octan-5-yl]propanoate |
NA |
270000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNLIP |
N'-[(2S)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]-N-(4-butoxyphenyl)butanediamide |
550000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNLIP |
N'-[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]-N-(4-butoxyphenyl)butanediamide |
170000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNLIP |
N'-[(1S)-2-[[(1S)-2-amino-1-naphthalen-2-yl-2-oxoethyl]amino]-1-naphthalen-2-yl-2-oxoethyl]-N-(4-butoxyphenyl)butanediamide |
360000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNLIP |
Koenimbine |
NA |
168600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNLIP |
methyl 2-[[(2E,8E)-deca-2,8-dienoyl]amino]-3-(5-hydroxy-6-oxo-3,8-dioxatricyclo[5.1.0.02,4]octan-5-yl)propanoate |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNMT |
3-(fluoromethyl)-N-(3-nitrophenyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide |
250000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNMT |
N-(3-chlorophenyl)-3-(fluoromethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide |
890000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNMT |
N-(4-nitrophenyl)-3-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNMT |
Thiopheneethanamine |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNMT |
alpha-(Aminomethyl)-3,4-dichlorobenzyl alcohol |
NA |
NA |
180000 |
NA |
NA |
NA |
BindingDB |
| PNMT |
9H-Fluorene-2-methanamine |
530000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNMT |
3-(Aminomethyl)thiophene |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |