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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PNP 593000 NA NA NA NA NA BindingDB
PNP 180000 NA NA NA NA NA BindingDB
PNP 270000 NA NA NA NA NA BindingDB
PNP 3-Benzylhypoxanthine NA 112000 NA NA NA NA BindingDB|TTD
PNP 4,7-Benzimidazoledione 550000|1650000 NA NA NA NA NA BindingDB|TTD
PNP 337000 NA NA NA NA NA BindingDB
PNP {Hydroxy-[5-(2-hydroxy-6-oxo-1,6-dihydro-purin-9-yl)-pentyl]-phosphinoylmethyl}-phosphonic acid 270000 NA NA NA NA NA BindingDB
PNP 110000 NA NA NA NA NA BindingDB
PNP 8-Amino-3-benzyl-1,9-dihydro-purine-6-thione NA 131000 NA NA NA NA BindingDB|TTD
PNP 1800000|2000000 NA NA NA NA NA BindingDB
PNP (2S,3S,4R,5S)-2-(4-amino-7H-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol NA 300000 NA NA NA NA BindingDB|TTD
PNP 2-amino-7-((2S,3S,4R,5S)-3,4-dihydroxy-5-(hydroxymethyl)tetrahydrofuran-2-yl)-3H-pyrrolo[2,3-d]pyrimidine-4(7H)-thione NA 315000 NA NA NA NA BindingDB|TTD
PNP 1-Benzylbenzimidazole-4,7-dione 580000|670000 NA NA NA NA NA BindingDB|TTD
PNP 1-[(4-Fluorophenyl)methyl]benzimidazole-4,7-dione 780000|990000 NA NA NA NA NA BindingDB|TTD
PNP 1-[(3-Fluorophenyl)methyl]benzimidazole-4,7-dione 520000|990000 NA NA NA NA NA BindingDB|TTD
PNP 1-[(2-Fluorophenyl)methyl]benzimidazole-4,7-dione 1480000|1500000 NA NA NA NA NA BindingDB|TTD
PNP 1-[(2-Methylthiazol-4-yl)methyl]benzimidazole-4,7-dione 110000 NA NA NA NA NA BindingDB
PNP 1-Methylbenzimidazole-4,7-dione 2210000 NA NA NA NA NA BindingDB|TTD
PNP 1-Butylbenzimidazole-4,7-dione 560000|2960000 NA NA NA NA NA BindingDB|TTD
PNP 1-Benzyl-2-methyl-benzimidazole-4,7-dione 300000|1050000 NA NA NA NA NA BindingDB|TTD