| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PNP |
1,2-Dibenzylbenzimidazole-4,7-dione |
350000|670000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PNP |
|
576000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PNP |
Adenosine |
2000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| PNP |
|
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB |
| PNP |
|
1500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PNP |
|
142000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PNP |
|
618000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PNP |
|
131000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PNP |
3-[(2S,3R,4S,5R)-3,4-dihydroxy-5-(hydroxymethyl)oxolan-2-yl]-1,7a-dihydropyrazolo[4,3-d]pyrimidin-7-one |
NA|110000 |
102000|NA |
NA |
NA |
NA |
NA |
BindingDB |
| PNP |
[(2R,3S,4R,5S)-3,4-dihydroxy-5-(7-oxo-1,7a-dihydropyrazolo[4,3-d]pyrimidin-3-yl)oxolan-2-yl]methyl 4-fluorosulfonylbenzoate |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PNP |
|
200000|290000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| POLA1 |
[[(2R,3R,5R)-5-(7-aminotriazolo[4,5-d]pyrimidin-3-yl)-3-hydroxyoxolan-2-yl]methoxy-(2,2-dimethylpropanoyloxymethoxy)phosphoryl]oxymethyl 2,2-dimethylpropanoate |
156000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| POLA1 |
[[(2R,3S,5R)-5-(6-amino-8-bromopurin-9-yl)-3-hydroxyoxolan-2-yl]methoxy-(2,2-dimethylpropanoyloxymethoxy)phosphoryl]oxymethyl 2,2-dimethylpropanoate |
548000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| POLA1 |
6H-Purin-6-one, 1,9-dihydro-2-((3-ethyl-4-methylphenyl)amino)- |
1760000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| POLA1 |
Gs-461203 |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB |
| POLA1 |
N-[[(2R,3R,5R)-5-(4-amino-2-oxopyrimidin-1-yl)-4,4-difluoro-3-hydroxyoxolan-2-yl]methoxy-hydroxyphosphinothioyl]benzamide |
NA |
NA |
NA |
350000 |
NA |
NA |
BindingDB|TTD |
| POLA1 |
|
1760000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| POLA1 |
2,2-Dimethyl-propionic acid [5-(7-amino-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl)-3-hydroxy-tetrahydro-furan-2-ylmethoxy]-(2,2-dimethyl-propionyloxymethoxy)-phosphoryloxymethyl ester |
156000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| POLA1 |
2-[(3S,10R,13R,17R)-17-((E)-(1R,4S)-4-Ethyl-1,5-dimethyl-hex-2-enyl)-10,13-dimethyl-2,3,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-3-yloxy]-ethanol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| POLA1 |
1-[(3S,10R,13R,17R)-17-((E)-(1R,4S)-4-Ethyl-1,5-dimethyl-hex-2-enyl)-10,13-dimethyl-2,3,4,7,8,9,10,11,12,13,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-3-yloxy]-ethane-1,2-diol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |