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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
POLB Stigmasterol NA 250000 NA NA NA NA PubChem
POLB Calanolide A NA 205000 NA NA NA NA BindingDB|PubChem
POLB 3-[7,7-Dimethyl-3-(2-methylbutanoyl)-4a,6-bis(3-methylbut-2-enyl)-2,4-dioxo-5,6-dihydrochromen-8-yl]hexanoic acid NA 342000 NA NA NA NA BindingDB
POLG 1-cyclopropyl-7-[4-(4-{4-[(3-ethyl-4-methylphenyl)amino]-2,6-dioxo-3,6-dihydropyrimidin-1(2H)-yl}butyl)-3-methylpiperazin-1-yl]-6,8-difluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acid 684000 NA NA NA NA NA BindingDB
POLH Montelukast Sodium NA NA NA NA 213313 NA PubChem
POLI Nonivamide NA NA NA NA 112202 NA PubChem
POLK N-Acetyl-L-Aspartic Acid NA NA NA NA 112202 NA PubChem
POLL 5-Hydroxy-3-Hydroxymethyl-2-Methyl-7-Methoxychromone NA 454000 NA NA NA NA BindingDB
POLL Mellein NA 316000 NA NA NA NA BindingDB
POLL Nodulisporol NA 168000 NA NA NA NA BindingDB
POLL 5-Formyl-8-Hydroxy-3-Methyl-3,4-Dihydroisocoumarin NA 275000 NA NA NA NA BindingDB
POLL 8-Methoxy-3-methylisochroman-1-one NA 180000 NA NA NA NA BindingDB
POLR2A 3'-Deoxycytidine 5'-triphosphate NA 500000 NA NA NA NA TTD
POLR2A Gs-461203 NA 500000 NA NA NA NA TTD
POLR2A 3-cyclohexyl-2-(furan-3-yl)-1H-indole-6-carboxylic acid NA 125000 NA NA NA NA TTD
POLR2A 3-cyclohexyl-2-furan-3-yl-1-methyl-1H-indole-6-carboxylic acid NA 125000 NA NA NA NA BindingDB|TTD
POLR2B 3'-Deoxycytidine 5'-triphosphate NA 500000 NA NA NA NA TTD
POLR2B Gs-461203 NA 500000 NA NA NA NA TTD
POLR2B 3-cyclohexyl-2-(furan-3-yl)-1H-indole-6-carboxylic acid NA 125000 NA NA NA NA TTD
POLR2B 3-cyclohexyl-2-furan-3-yl-1-methyl-1H-indole-6-carboxylic acid NA 125000 NA NA NA NA TTD