| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| POLR2C |
3'-Deoxycytidine 5'-triphosphate |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| POLR2C |
Gs-461203 |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| POLR2C |
3-cyclohexyl-2-(furan-3-yl)-1H-indole-6-carboxylic acid |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| POLR2C |
3-cyclohexyl-2-furan-3-yl-1-methyl-1H-indole-6-carboxylic acid |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| PON1 |
2-[(2,3-dimethylimidazol-3-ium-1-yl)methyl]-1H-benzimidazole;chloride |
NA |
625710 |
NA |
NA |
NA |
NA |
TTD |
| PON1 |
4-[(2,3-Dimethylimidazol-3-ium-1-yl)methyl]-5,7-dimethylchromen-2-one;chloride |
NA |
317310 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PON1 |
1-[(3-Butylbenzimidazol-1-ium-1-yl)methyl]benzotriazole;chloride |
NA |
3333300 |
NA |
NA |
NA |
NA |
TTD |
| PON1 |
1-[(3-Benzylbenzimidazol-1-ium-1-yl)methyl]benzotriazole;chloride |
NA |
2064200 |
NA |
NA |
NA |
NA |
TTD |
| PON1 |
4-[[3-(Benzotriazol-1-ylmethyl)benzimidazol-3-ium-1-yl]methyl]-7,8-dimethylchromen-2-one;chloride |
NA |
237500 |
NA |
NA |
NA |
NA |
TTD |
| PON1 |
4-[[3-(Benzotriazol-1-ylmethyl)benzimidazol-3-ium-1-yl]methyl]-6-tert-butylchromen-2-one;chloride |
NA |
627000 |
NA |
NA |
NA |
NA |
TTD |
| PON1 |
Phenylphosphate |
NA |
3250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PON1 |
(2-Bromo-4,5-dihydroxyphenyl)(2,3-dibromo-5,6-dihydroxyphenyl)methanone (11) |
NA |
1110000 |
NA |
NA |
NA |
NA |
BindingDB |
| PON1 |
Docetaxel |
291000 |
665000 |
NA |
NA |
NA |
NA |
BindingDB |
| PON1 |
2-Hydroxy-4-[(E)-{4-[(pyridin-2-yl)sulfamoyl]phenyl}diazenyl]benzoic acid |
570000 |
260000 |
NA |
NA |
NA |
NA |
BindingDB |
| PON1 |
2-amino-4,5-dimethoxy-N-pyridin-2-ylbenzamide |
NA |
237500 |
NA |
NA |
NA |
NA |
BindingDB |
| PON1 |
Diethyl phenyl phosphate |
NA |
3270000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PON1 |
Phosphoric acid, p-aminophenyl diethyl ester |
NA |
1280000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PON1 |
Acetazolamide |
743000 |
800000 |
NA |
NA |
NA |
NA |
BindingDB |
| PON1 |
2,3,3',4'-Tetramethoxybenzophenone |
NA |
1212000 |
NA |
NA |
NA |
NA |
BindingDB |
| PON1 |
Lincomycin |
18300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |