| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PON1 |
(3-Bromo-4,5-dimethoxyphenyl)(2,3-dibromo-5,6-dimethoxyphenyl)methanone (9) |
NA |
125000 |
NA |
NA |
NA |
NA |
BindingDB |
| PON1 |
(2,3-Dibromo-5,6-dihydroxyphenyl)(3,4-dihydroxyphenyl)methanone (10) |
NA |
832000 |
NA |
NA |
NA |
NA |
BindingDB |
| PON1 |
(3-Bromo-4,5-dihydroxyphenyl)(2,3-dibromo-5,6-dihydroxyphenyl)methanone (12) |
NA |
701000 |
NA |
NA |
NA |
NA |
BindingDB |
| PON1 |
Desacetyl acetazolamide |
2001000 |
1240000 |
NA |
NA |
NA |
NA |
BindingDB |
| PON1 |
Netilmycin sulfate |
3730000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| POU3F2 |
N-(3-fluorophenyl)-4-[2-(4-hydroxyanilino)-2-oxoethoxy]naphthalene-1-carboxamide |
NA |
138000 |
NA |
NA |
NA |
NA |
BindingDB |
| POU3F2 |
N-(3-fluorophenyl)-4-[2-(3-hydroxyanilino)-2-oxoethoxy]naphthalene-1-carboxamide |
NA |
148000 |
NA |
NA |
NA |
NA |
BindingDB |
| POU3F2 |
4-[(2,2,2-Trifluoro-ethylcarbamoyl)-methoxy]-naphthalene-1-carboxylic acid (3-fluoro-phenyl)-amide |
NA |
204000 |
NA |
NA |
NA |
NA |
BindingDB |
| POU3F3 |
N-(3-fluorophenyl)-4-[2-(4-hydroxyanilino)-2-oxoethoxy]naphthalene-1-carboxamide |
NA |
124000 |
NA |
NA |
NA |
NA |
BindingDB |
| POU3F3 |
4-Cyclopropylcarbamoylmethoxy-naphthalene-1-carboxylic acid (3-fluoro-phenyl)-amide |
NA |
810000 |
NA |
NA |
NA |
NA |
BindingDB |
| POU3F3 |
N-(3-fluorophenyl)-4-[2-(3-hydroxyanilino)-2-oxoethoxy]naphthalene-1-carboxamide |
NA |
142000 |
NA |
NA |
NA |
NA |
BindingDB |
| POU3F3 |
4-[(2,2,2-Trifluoro-ethylcarbamoyl)-methoxy]-naphthalene-1-carboxylic acid (3-fluoro-phenyl)-amide |
NA |
162000 |
NA |
NA |
NA |
NA |
BindingDB |
| PPARA |
N-(4-acetamidophenyl)sulfonyl-2-[(5-chloro-1,3-benzothiazol-2-yl)sulfanyl]pentanamide |
NA |
108000 |
NA |
NA |
NA |
NA |
TTD |
| PPARA |
2,2-dimethyl-5-[4-[(E)-2-pyridin-4-ylethenyl]phenoxy]pentanoic acid |
NA |
NA |
NA |
103200 |
NA |
NA |
TTD |
| PPARA |
N-octadecylsulfamide |
NA |
NA |
NA |
10000000 |
NA |
NA |
TTD |
| PPARA |
N-hexadecylsulfamide |
NA |
NA |
NA |
10000000 |
NA |
NA |
TTD |
| PPARA |
N-(2-adamantyl)-N'-propylsulfamide |
NA |
NA |
NA |
10000000 |
NA |
NA |
TTD |
| PPARA |
2-[(1S)-5-[3-(2-propyl-4-{5H,6H,7H-pyrano[2,3-d][1,3]thiazol-2-yl}phenoxy)propoxy]-2,3-dihydro-1H-inden-1-yl]acetic acid |
NA |
NA |
NA |
9901477.39 |
NA |
NA |
TTD |
| PPARA |
Gemfibrozil |
NA |
NA |
NA |
193300|15190000 |
NA |
NA |
PubChem |
| PPARA |
3-(((6-((5-Cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid |
NA |
NA |
NA |
680000 |
NA |
NA |
TTD |