Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| PON1 | Solaraze | 805000 | 1639000 | NA | NA | NA | NA | BindingDB |
| PON1 | Furosemide [USAN:USP:INN:BAN:JAN] | 702000 | 360000 | NA | NA | NA | NA | BindingDB |
| PON1 | Etoposide | 131000 | 226000 | NA | NA | NA | NA | BindingDB |
| PON1 | Ifosfamide | 8973000 | 23300000 | NA | NA | NA | NA | BindingDB |
| PON1 | 4-Nitrophenyl Phosphate | NA | 18500000 | NA | NA | NA | NA | BindingDB|TTD |
| PON1 | Ketoprofen | 13010000 | 6230000 | NA | NA | NA | NA | BindingDB |
| PON1 | Lincomycin A | 11116000 | 13010000 | NA | NA | NA | NA | BindingDB |
| PON1 | Mafenide | 340000 | 190000 | NA | NA | NA | NA | BindingDB |
| PON1 | 2-amino-N'-(3-chlorophenyl)-4,5-dimethoxybenzenecarboximidamide | NA | 627000 | NA | NA | NA | NA | BindingDB |
| PON1 | NA | 3333300 | NA | NA | NA | NA | BindingDB | |
| PON1 | NA | 564130 | NA | NA | NA | NA | BindingDB | |
| PON1 | NA | 625710 | NA | NA | NA | NA | BindingDB | |
| PON1 | NA | 2064200 | NA | NA | NA | NA | BindingDB | |
| PON1 | Clindamycin Phosphate | 35800000 | NA | NA | NA | NA | NA | BindingDB |
| PON1 | Oxytetracycline | 200000 | NA | NA | NA | NA | NA | BindingDB |
| PON1 | Tenoxicam | 306000 | 340000 | NA | NA | NA | NA | BindingDB |
| PON1 | 2-[(1S,2R,3R,4S,5R,6R)-2-[(2S,3S,4S,5R)-3-[(2R,3R,4R,5S,6R)-4,5-dihydroxy-6-(hydroxymethyl)-3-(methylamino)tetrahydropyran-2-yl]oxy-4-formyl-4-hydroxy-5-methyl-tetrahydrofuran-2-yl]oxy-5-guanidino-3,4,6-trihydroxy-cyclohexyl]guanidine | 56300000 | NA | NA | NA | NA | NA | BindingDB |
| PON1 | 1-(1H-benzimidazol-1-ylmethyl)-1H-1,2,3-benzotriazole | NA | 564130 | NA | NA | NA | NA | TTD |
| PON1 | (2,3-Dibromo-5,6-dimethoxyphenyl)(3,4-dimethoxyphenyl)methanone (7) | NA | 174000 | NA | NA | NA | NA | BindingDB |
| PON1 | (2-Bromo-4,5-dimethoxyphenyl)(2,3-dibromo-5,6-dimethoxyphenyl)methanone (8) | NA | 123000 | NA | NA | NA | NA | BindingDB |