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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLG N-[[4-(diaminomethylideneamino)phenyl]methyl]-4-[7-[4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazin-1-yl]-7-oxoheptanoyl]piperazine-1-carboxamide 1000000 NA NA NA NA NA TTD
PLG N-[[4-(diaminomethylideneamino)phenyl]methyl]-4-[6-[4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazin-1-yl]-6-oxohexanoyl]piperazine-1-carboxamide 316000 NA NA NA NA NA BindingDB|TTD
PLG [2-(4-Guanidino-benzylcarbamoyl)-ethyl]-carbamic acid 4-[2-(4-guanidino-benzylcarbamoyl)-ethylcarbamoyloxymethyl]-benzyl ester 1000000 NA NA NA NA NA TTD
PLG [(4-Guanidino-benzylcarbamoyl)-methyl]-carbamic acid 4-[(4-guanidino-benzylcarbamoyl)-methylcarbamoyloxymethyl]-benzyl ester 1000000 NA NA NA NA NA TTD
PLG [5-[4-(Benzylcarbamoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(benzylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG N'-[[4-(diaminomethylideneamino)phenyl]methyl]-N-[[4-[[[4-[[4-(diaminomethylideneamino)phenyl]methylamino]-4-oxobutanoyl]amino]methyl]phenyl]methyl]butanediamide 1000000 NA NA NA NA NA TTD
PLG N-[[4-(diaminomethylideneamino)phenyl]methyl]-4-[9-[4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazin-1-yl]-9-oxononanoyl]piperazine-1-carboxamide 1000000 NA NA NA NA NA TTD
PLG Pentanedioic acid 4-aminomethyl-benzylamide 4-{[4-(4-aminomethyl-benzylcarbamoyl)-butyrylamino]-methyl}-benzylamide 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(4-imidazol-1-ylbutanoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[3-(2-aminopyrimidin-5-yl)propanoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[3-(6-aminopyridin-3-yl)propanoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(3-pyridin-4-ylsulfanylpropanoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-(2-Piperidin-4-ylethylcarbamoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(2-piperidin-4-ylethylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[2-[4-(2-Aminoethyl)phenyl]ethylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-[4-(2-aminoethyl)phenyl]ethylcarbamoyl]piperazine-1-carboxylate 570000 NA NA NA NA NA BindingDB|TTD
PLG [5-[4-[[4-(Methylaminomethyl)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[[4-(methylaminomethyl)phenyl]methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[3-(pyridin-4-ylamino)propanoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(6-imidazol-1-ylhexanoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [(R)-1-(4-Aminomethyl-benzylcarbamoyl)-ethyl]-carbamic acid 4-[(R)-1-(4-aminomethyl-benzylcarbamoyl)-ethylcarbamoyloxymethyl]-benzyl ester 1000000 NA NA NA NA NA TTD
PLG [(4-Aminomethyl-benzylcarbamoyl)-methyl]-methyl-carbamic acid 4-({[(4-aminomethyl-benzylcarbamoyl)-methyl]-methyl-carbamoyloxy}-methyl)-benzyl ester 230000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[(4-aminophenyl)methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD