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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PLG [4-[[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxymethyl]cyclohexyl]methyl 4-[[4-(diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[2-(1-Carbamimidoylpiperidin-4-yl)acetyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-(1-carbamimidoylpiperidin-4-yl)acetyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[2-(1-Carbamimidoylpiperidin-4-yl)ethylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-(1-carbamimidoylpiperidin-4-yl)ethylcarbamoyl]piperazine-1-carboxylate 632000 NA NA NA NA NA BindingDB|TTD
PLG [5-[4-[3-(1-Carbamimidoylpiperidin-4-yl)propanoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[3-(1-carbamimidoylpiperidin-4-yl)propanoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[3-[4-(Diaminomethylideneamino)phenyl]propanoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[3-[4-(diaminomethylideneamino)phenyl]propanoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[2-[4-(2-Aminoethyl)phenyl]acetyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-[4-(2-aminoethyl)phenyl]acetyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG 1,5-Di{4-[4-amino(imino)methylbenzylcarbamoyl]hexahydro-1-pyrazinylcarbonyloxy}cyclooctane 134000 NA NA NA NA NA BindingDB|TTD
PLG [5-[4-(4-Aminobutylcarbamoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(4-aminobutylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Aminomethyl)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[[4-(aminomethyl)phenyl]methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[2-[4-(Diaminomethylideneamino)phenyl]acetyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[2-[4-(diaminomethylideneamino)phenyl]acetyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-(5-Aminopentylcarbamoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(5-aminopentylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-(6-Aminohexylcarbamoyl)piperazine-1-carbonyl]oxycyclooctyl] 4-(6-aminohexylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(5-aminopentylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[(1-Carbamimidoylpiperidin-4-yl)methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-[(1-carbamimidoylpiperidin-4-yl)methylcarbamoyl]piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG 1-Methyl-1H-indole-5-carboximidamide 1000000 NA NA NA NA NA TTD
PLG 4-Chloro-N-(2-{3-[2-(pyridin-4-ylamino)-ethoxy]-phenyl}-ethyl)-benzenesulfonamide 500000 NA NA NA NA NA TTD
PLG m-Aminobenzamidine hydrochloride 125000 NA NA NA NA NA BindingDB
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(4-aminobutylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG [5-[4-[[4-(Diaminomethylideneamino)phenyl]methylcarbamoyl]piperazine-1-carbonyl]oxycyclooctyl] 4-(3-aminopropylcarbamoyl)piperazine-1-carboxylate 1000000 NA NA NA NA NA TTD
PLG Benzamidine 350000|500000|2510000 NA NA NA NA NA BindingDB|TTD