| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PLG |
N-[(1S)-5-amino-1-cyanopentyl]-7-methyl-6-[[3-[3-(2-methylpropyl)-2-oxo-1,3-benzoxazol-6-yl]-2,5-dioxoimidazolidin-1-yl]methyl]pyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
N-[(1S)-5-amino-1-cyanopentyl]-6-[[2,5-dioxo-3-[2-oxo-3-(pyridin-4-ylmethyl)-1,3-benzoxazol-6-yl]imidazolidin-1-yl]methyl]-7-methylpyrrolo[2,3-d]pyrimidine-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
N-[(1S)-5-amino-1-cyanopentyl]-5-[[3-(4-fluorophenyl)-2,5-dioxoimidazolidin-1-yl]methyl]-1,3-benzoxazole-2-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
N-[(1S)-5-amino-1-cyanopentyl]-2-[[2,5-dioxo-3-(4-phenoxyphenyl)imidazolidin-1-yl]methyl]-1-methylbenzimidazole-5-carboxamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
3-(Phenylmethyl)benzenecarboximidamide |
3160000|125892.54 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
5-Amidinoindole |
112000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
3-Nitrobenzamidinium hydrochloride |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
2-[4-[[(2S)-2-[[4-(aminomethyl)cyclohexanecarbonyl]amino]-3-phenylpropanoyl]amino]phenyl]acetic acid |
NA |
620000 |
NA |
NA |
NA |
NA |
BindingDB |
| PLG |
(3R,8R,11S,14S,17S,20S,23S,26S,29S,32S)-3-amino-20-[(1-carbamimidoylpiperidin-4-yl)methyl]-11-(carboxymethyl)-23-(hydroxymethyl)-17,26-bis[(4-hydroxyphenyl)methyl]-29-methyl-14-(2-methylpropyl)-2,10,13,16,19,22,25,28,31-nonaoxo-5,6-dithia-1,9,12,15,18,21,24,27,30-nonazabicyclo[30.3.0]pentatriacontane-8-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PLG |
H-D-Ser-Ala-Arg-NH-(CH2)6-NH2 (5) |
181000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLG |
H-D-Ser-Ala-Arg-NH-(CH2)7-NH2 (6) |
364000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLG |
H-D-Ser-Ala-Arg-NH-(CH2)2-OH (9) |
727000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLG |
H-D-Ser-Ala-Arg-NH-(CH2)3-OH (10) |
1090000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLG |
H-D-Ser-Ala-Arg-NH-(CH2)4-OH (11) |
545000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PLG |
N-[(6-amino-2-methylpyridin-3-yl)methyl]-1-[[4-(pyrazol-1-ylmethyl)phenyl]methyl]pyrazole-4-carboxamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
ASGPR modulator-1 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
(8e)-3-Amino-1-Methyl-15-[(1h-Pyrazol-1-Yl)methyl]-7,10,11,12,24,25-Hexahydro-6h,18h,23h-19,22-(Metheno)pyrido[4,3-J][1,9,13,17,18]benzodioxatriazacyclohenicosin-23-One |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
1-(4-Amidinobenzyl)indole |
111000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PLG |
2-[[6-amino-5-[(Z)-N'-hydroxycarbamimidoyl]pyrazin-2-yl]amino]acetic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| PLG |
benzyl 2-[[6-amino-3-chloro-5-[(Z)-N'-hydroxycarbamimidoyl]pyrazin-2-yl]amino]acetate |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |