| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PRKACB |
2-[5,6-Bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKACB |
Harmine |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKACB |
Alvocidib |
NA |
960000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKACB |
Imatinib |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKACG |
Roscovitine |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKACG |
2-[5,6-Bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKACG |
Harmine |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKACG |
Alvocidib |
NA |
960000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKACG |
Imatinib |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKCA |
5,5'-(1E)-1,2-Ethenediylbis-1,2,3-benzenetriol |
NA |
NA |
NA |
2980000 |
NA |
NA |
BindingDB|TTD |
| PRKCA |
N-Decyl-4-aminoquinaldinium iodide |
NA |
117000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PRKCA |
[(2R,3R,4R,5R,6R)-5-hydroxy-6-[2-(3-hydroxy-4-methoxyphenyl)ethoxy]-4-[(2R,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxy-2-[[(2R,3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxymethyl]oxan-3-yl] (E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enoate |
NA |
125000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PRKCA |
2-(2-Methyl-5-nitroanilino)-4-(3-pyridyl)pyrimidine |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCA |
7-(4-fluoroanilino)-1-[(1R,3R)-3-hydroxycyclopentyl]-3-(4-methoxyphenyl)-4H-pyrimido[4,5-d]pyrimidin-2-one |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| PRKCA |
(2S,5S)-5-Hydroxymethyl-2-isopropyl-1-methyl-1,2,4,5-tetrahydro-benzo[e][1,4]diazepin-3-one |
127000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PRKCA |
1-Methyl-4-amino-2-methylquinolinium |
NA |
3590000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PRKCA |
3-[(2R,4R,5S,6R)-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]-13-(1,3-dihydroxypropan-2-ylamino)-6,20-dihydroxy-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaene-12,14-dione |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| PRKCA |
3-[(2S,4R,5S,6R)-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]-13-(1,3-dihydroxypropan-2-ylamino)-6,20-dihydroxy-3,13,23-triazahexacyclo[14.7.0.02,10.04,9.011,15.017,22]tricosa-1,4(9),5,7,10,15,17(22),18,20-nonaene-12,14-dione |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| PRKCA |
Tetradecanoic acid (2R,3R)-2-hydroxymethyl-5-oxo-tetrahydro-furan-3-yl ester |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PRKCA |
4-(4-Morpholinylamino)benzoic acid |
NA |
188000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |