| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PREP |
Boldine 2-methyl ether |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB |
| PREP |
(2R)-4-(2-Benzoyl-1,2-diazepan-1-YL)-4-oxo-1-(2,4,5-trifluorophenyl)butan-2-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| PREP |
Palmatine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PREP |
Berberine |
NA |
142000|145000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PREP |
Berbamine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PREP |
Aromoline |
NA |
189000 |
NA |
NA |
NA |
NA |
TTD |
| PREP |
Obamegine |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PREP |
Rutin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PREP |
Kaempferol |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PREP |
3,7-Dihydroxyflavone |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PREP |
Vildagliptin |
NA |
210000 |
NA |
NA |
NA |
NA |
BindingDB |
| PREP |
Galantamine |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PRKAB1 |
2-[4-(1,2-Dihydroimidazo[1,2-a]benzimidazol-4-ylmethyl)phenyl]benzonitrile;hydrobromide |
NA |
NA |
NA |
109000 |
NA |
NA |
BindingDB |
| PRKACA |
[3-(2-Imidazol-1-yl-ethoxy)-phenyl]-(4-pyridin-3-yl-pyrimidin-2-yl)-amine |
NA |
340000 |
NA |
NA |
NA |
NA |
BindingDB |
| PRKACA |
|
NA |
171719 |
NA |
NA |
NA |
NA |
BindingDB |
| PRKACA |
(3RS,4R)-4-{9-Isopropyl-6-[(pyridin-3-ylmethyl)-amino]-9H-purin-2-ylamino}-2-methyl-hexan-3-ol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| PRKACA |
Roscovitine |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKACA |
2-[5,6-Bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem |
| PRKACA |
2-N-(2-aminoethyl)-9-ethyl-6-N-[3-(trifluoromethyl)phenyl]purine-2,6-diamine |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB |
| PRKACA |
(1S,3R,4R)-methyl 3-(6-amino-9H-purin-9-yl)-4-hydroxycyclopentanecarboxylate |
NA |
168000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |