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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PRMT1 1-Hydroxy-6-amino-3-naphthalenesulfonic acid NA 928000 NA NA NA NA TTD
PRMT1 1-Naphthol-8-amino-3,6-disulfonic acid NA 540000 NA NA NA NA TTD
PRMT1 fluorone Black NA 126000 NA NA NA NA TTD
PRMT1 (r)-2-Amino-n-ethyl-propanamide NA 1000000 NA NA NA NA TTD
PRMT3 N-[3-[4-[[2-hydroxyethyl(methyl)amino]methyl]-1H-pyrrol-3-yl]phenyl]prop-2-enamide NA 200000 NA NA NA NA TTD
PRMT3 Methyl(2-(4-methylpiperidin-1-yl)ethyl)amine NA 500000 NA NA NA NA TTD
PRMT3 (r)-2-Amino-n-ethyl-propanamide NA 1000000 NA NA NA NA TTD
PRMT5 5-[5-(4-Carbamimidoylphenyl)furan-2-yl]pyridine-2-carboximidamide NA 186000 NA NA NA NA TTD
PRMT5 Furamidine NA 166000|256000 NA NA NA NA PubChem|TTD
PRMT5 (2S)-6-amino-2-[[(2S)-2-[[2-[[2-[[(2S)-6-amino-2-[[2-[[(2S)-2-[[2-[[(2S)-6-amino-2-[[2-[[2-[[5-[(1-amino-2-chloroethylidene)amino]-2-[[(2S)-2-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-(hex-5-ynoylamino)-3-(1H-imidazol-5-yl)propanoyl]amino]hexanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]pentanoyl]amino]acetyl]amino]acetyl]amino]hexanoyl]amino]acetyl]amino]-4-methylpentanoyl]amino]acetyl]amino]hexanoyl]amino]acetyl]amino]acetyl]amino]propanoyl]amino]hexanoic acid NA 500000 NA NA NA NA TTD
PRMT5 4-(aminomethyl)-6-(1-methylpyrazol-4-yl)-2H-phthalazin-1-one NA NA 110000 NA NA NA ChEMBL
PRMT5 Pentamidine NA 582000 NA NA NA NA PubChem|TTD
PRMT5 Stilbamidine NA 712000 NA NA NA NA TTD
PRMT5 Hexamidine NA 357000 NA NA NA NA PubChem|TTD
PRMT6 Furamidine NA 283000 NA NA NA NA PubChem
PRMT6 N-Methyl-N-(3-thien-2-ylbenzyl)amine NA 125000 NA NA NA NA ChEMBL
PRMT6 N-[3-(2-Furyl)benzyl]-N-methylamine NA 146000 NA NA NA NA ChEMBL
PRMT6 [3-(Pyrrolidin-1-ylmethyl)phenyl]methanamine NA 360000 NA NA NA NA ChEMBL
PRMT6 Sulfathiazole NA 430000 NA NA NA NA ChEMBL|PubChem
PRMT6 N-Methyl-N-[3-(2-methyl-1,3-thiazol-4-YL)benzyl]amine NA 136000 NA NA NA NA ChEMBL