| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PROC |
N-[4-Guanidino-1-(thiazole-2-carbonyl)-butyl]-2-[2-oxo-4-(quinoline-8-sulfonyl)-piperazin-1-yl]-acetamide |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| PROC |
N-[(R)-4-Guanidino-1-(thiazole-2-carbonyl)-butyl]-2-(2-oxo-4-phenylmethanesulfonyl-piperazin-1-yl)-acetamide |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| PROC |
N-[(2S)-6-amino-1-[5-[[4-[2-(3,4-dichlorophenyl)ethoxy]phenyl]methyl]-1,2,4-oxadiazol-3-yl]-1-oxohexan-2-yl]-3,4-difluorobenzamide |
150000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| PROC |
(9R,12S)-19-chloro-9-cyclohexyl-12-(2-methylpropyl)-8,11,14,23-tetrazatricyclo[14.7.0.017,22]tricosa-1(16),17(22),18,20-tetraene-7,10,13-trione |
NA |
395300 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PROC |
N-((R)-2-((S)-1-((2-allyl-5-chloro-1H-indol-3-yl)methylamino)-4-methyl-1-oxopentan-2-ylamino)-1-cyclohexyl-2-oxoethyl)pent-4-enamide |
NA |
284100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PROC |
(S)-N-((R)-2-((S)-1-((2-allyl-5-chloro-1H-indol-3-yl)methylamino)-4-methyl-1-oxopentan-2-ylamino)-1-cyclohexyl-2-oxoethyl)-2-phenylpent-4-enamide |
NA |
103500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PROC |
(3E,6S,9R,12S)-19-chloro-9-cyclohexyl-12-(2-methylpropyl)-6-phenyl-8,11,14,23-tetrazatricyclo[14.7.0.017,22]tricosa-1(16),3,17(22),18,20-pentaene-7,10,13-trione |
NA |
144500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PROC |
2''-Sulfamoyl-biphenyl-4-carboxylic acid [2-(3-carbamimidoyl-phenoxy)-phenyl]-amide |
NA |
181000 |
NA |
NA |
NA |
NA |
TTD |
| PRPS1 |
Phosphoric acid mono-[(2R,3R,4S,5R)-5-(6-amino-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-ylmethyl] ester |
NA |
5100000 |
NA |
NA |
NA |
NA |
BindingDB |
| PRPS1 |
{2-[(1R,3S)-3-(6-Amino-purin-9-yl)-cyclopentyl]-1,1-difluoro-ethyl}-phosphonic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| PRPS1 |
2-[(1R,3S)-3-(6-aminopurin-9-yl)cyclopentyl]ethyl dihydrogen phosphate |
NA |
600000 |
NA |
NA |
NA |
NA |
BindingDB |
| PRPS1 |
Adefovir |
NA |
3200000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PRPSAP2 |
2-(6-aminopurin-7-yl)ethoxymethyl-[(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(phosphonooxymethyl)oxolan-3-yl]oxyphosphinic acid |
790000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PRPSAP2 |
7-[2-(Phosphonomethoxy)ethyl]adenine |
17000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PRPSAP2 |
Adefovir |
3000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| PRSS1 |
Phenethylamine |
NA |
NA |
10964782 |
NA |
NA |
NA |
BindingDB |
| PRSS1 |
2-pyridin-2-yl-1H-benzimidazole-6-carboximidamide |
101000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| PRSS1 |
2-[6-Methyl-2-oxo-3-(2-pyridin-2-yl-ethylamino)-2H-pyrazin-1-yl]-N-(1H-pyrrolo[2,3-b]pyridin-5-ylmethyl)-acetamide |
140000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PRSS1 |
2-[6-Methyl-2-oxo-3-(2-pyridin-2-yl-ethylamino)-2H-pyrazin-1-yl]-N-(1H-pyrrolo[2,3-c]pyridin-5-ylmethyl)-acetamide |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| PRSS1 |
(2S)-1-[(2R)-2-amino-3,3-diphenylpropanoyl]-N-(4,5,6,7-tetrahydro-1H-indazol-5-ylmethyl)pyrrolidine-2-carboxamide |
216600 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |