| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTGS1 |
Sodium;2-[2-(2,6-dichloroanilino)-6-hydroxyphenyl]acetate |
NA |
4677351.41 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
Sodium;2-[2-(2,6-dichloroanilino)-5-fluorophenyl]acetate |
NA |
741310241.3 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
Sodium;2-[2-(2,6-dichloro-4-fluoroanilino)phenyl]acetate |
NA |
891250938.1 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
Sodium;2-[2-(2,6-dichloro-4-fluoroanilino)-5-fluorophenyl]acetate |
NA |
562341325.2 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
2-[(4-Cyclohexylpiperazin-1-yl)methyl]-4,6-dimethyl-[1,2]thiazolo[5,4-b]pyridin-3-one |
NA |
660693.45 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
Celecoxib |
NA |
12530000 |
NA |
NA |
NA |
NA |
PubChem |
| PTGS1 |
5-Hydroxydiclofenac |
NA |
446684|446683.59 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PTGS1 |
4',5-Dihydroxydiclofenac |
NA |
912010.84 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
3-Methoxyacetaminophen |
NA |
234000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
Atractylon |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-(Benzylideneamino)benzenesulfonamide |
NA |
108340 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-((4-(Dimethylamino)benzylidene)amino)benzenesulfonamide |
NA |
195740 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
Salicylic Acid |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| PTGS1 |
4-(4-Hydroxybenzylideneamino)benzenesulfonamide |
NA |
148200 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-[(3,5-Trimethoxy-benzylidene)-amino]-benzenesulfonamide |
NA |
167090 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-[(3,5-Dimethoxy-benzylidene)-amino]-benzenesulfonamide |
NA |
109690 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-[(3,4-Dimethoxy-benzylidene)-amino]-benzenesulfonamide |
NA |
110270 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-[(4-Fluorobenzylidene)amino]benzenesulfonamide |
NA |
159070 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-[(4-Trifluoromethyl-benzylidene)-amino]-benzenesulfonamide |
NA |
182190 |
NA |
NA |
NA |
NA |
TTD |
| PTGS1 |
4-[(4-Sulfamoyl-phenylimino)-methyl]-benzoic acid methyl ester |
NA |
183500 |
NA |
NA |
NA |
NA |
TTD |