Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTGS1 [5-(4-Methanesulfonyl-phenyl)-2-methyl-1-phenyl-1H-pyrrol-3-yl]-acetic acid NA 132000 NA NA NA NA TTD
PTGS1 3-(3,5-Dihydroxyphenyl)-6,8-dihydroxy-2H-1-benzopyran-2-one NA 285000 NA NA NA NA TTD
PTGS1 3-(3,5-Dimethoxyphenyl)-7-hydroxy-2H-1-benzopyran-2-one NA 105000 NA NA NA NA TTD
PTGS1 4-(dimethylamino)-2-methyl-5-(3-oxo-3-phenylprop-1-enyl)pyridazin-3(2H)-one NA 221300 NA NA NA NA TTD
PTGS1 (E)-2-methyl-5-(3-oxo-3-phenylprop-1-enyl)-6-phenylpyridazin-3(2H)-one NA 150000 NA NA NA NA TTD
PTGS1 Resveratrol NA 195500 NA NA NA NA PubChem
PTGS1 ((m-tolylimino)methyl)-4H-chromen-4-one NA 1000000 NA NA NA NA TTD
PTGS1 (E)-2-((4-oxo-4H-chromen-3-yl)methyleneamino)benzoic acid NA 1000000 NA NA NA NA TTD
PTGS1 Ballotetroside NA 1000000 NA NA NA NA TTD
PTGS1 2-(6-Chloro-9H-carbazol-2-yl)-propionic acid 2-nitrooxy-ethyl ester NA 110000 NA NA NA NA TTD
PTGS1 2-(6-Chloro-9H-carbazol-2-yl)-propionic acid 2-nitrooxy-propyl ester NA 123000 NA NA NA NA TTD
PTGS1 2-Methyl-5-[4-(methylsulfonyl)phenyl]-1-[3-(fluoro)phenyl]-1H-pyrrol-3-acetic acid NA 125000 NA NA NA NA TTD
PTGS1 2-[3-[4-(3-Chlorophenyl)piperazin-1-yl]propyl]-4,6-dimethyl-isothiazolo[5,4-b]pyridin-3-one NA 524807.46 NA NA NA NA TTD
PTGS1 N-Sinapoyl Serotonin NA 400000 NA NA NA NA TTD
PTGS1 8-Fluoro-2-{3-[3-fluoro-5-(4-methoxytetrahydro-4H-4-pyranyl)phenoxy]propyl}-5-(4-methanesulfonylbenzyl)-2,3,4,5-tetrahydro-1H-pyrido[4,3-b]indole hydrochloride NA 180300 NA NA NA NA TTD
PTGS1 N''-((4-oxo-4H-chromen-3-yl)methylene)butyrohydrazide NA 1000000 NA NA NA NA TTD
PTGS1 Rofecoxib NA 500000|159700 NA NA NA NA PubChem
PTGS1 Serotonin NA 400000 NA NA NA NA PubChem|TTD
PTGS1 Fraxetin NA 524000 NA NA NA NA TTD
PTGS1 Daphnetin NA 140000 NA NA NA NA PubChem|TTD