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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTGS1 Butein NA 120000 NA NA NA NA TTD
PTGS1 Atractylenolide I NA 200000 NA NA NA NA TTD
PTGS1 Sodium;2-[2-(4-hydroxyphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 326000 NA NA NA NA TTD
PTGS1 2-[1-(4-Chlorobenzoyl)-2-ethylindol-3-yl]acetic acid NA 400000 NA NA NA NA TTD
PTGS1 Sulfinpyrazone NA 509100 NA NA NA NA PubChem
PTGS1 Piroxicam NA 254600 NA NA NA NA PubChem
PTGS1 N-[4-[2-(3,4-dichlorophenyl)ethyl]phenyl]-4-hydroxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide NA 489000 NA NA NA NA TTD
PTGS1 N-(3',4'-Dichloro[1,1'-biphenyl]-4-yl)-4-hydroxy-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide NA 118000 NA NA NA NA TTD
PTGS1 4-(4-Nitro-benzylideneamino)-benzenesulfonamide NA 141250 NA NA NA NA TTD
PTGS1 Disodium;4-[5-(1-carboxylatoethyl)-2-[(2-oxocyclopentyl)methyl]phenyl]benzoate NA 1000000 NA NA NA NA TTD
PTGS1 Sodium;2-[4-[(2-oxocyclopentyl)methyl]-2-phenylphenyl]propanoate NA 310000 NA NA NA NA TTD
PTGS1 Sodium;2-[4-[(2-oxocyclopentyl)methyl]-2-[4-(trifluoromethoxy)phenyl]phenyl]propanoate NA 515000 NA NA NA NA TTD
PTGS1 Sodium;2-[2-iodo-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 270000 NA NA NA NA TTD
PTGS1 Sodium;2-[3-(4-methoxyphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 800000 NA NA NA NA TTD
PTGS1 Sodium;2-[3-(4-fluorophenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 174000 NA NA NA NA TTD
PTGS1 Sodium;2-[2-(4-methylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 470000 NA NA NA NA TTD
PTGS1 Sodium;2-[3-(4-hydroxyphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 1000000 NA NA NA NA TTD
PTGS1 Sodium;2-[2-(4-methylsulfanylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 575000 NA NA NA NA TTD
PTGS1 Sodium;2-[2-(4-fluorophenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 174000 NA NA NA NA TTD
PTGS1 Disodium;4-[2-(1-carboxylatoethyl)-5-[(2-oxocyclopentyl)methyl]phenyl]benzoate NA 1000000 NA NA NA NA TTD