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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTGS1 Sodium;2-[4-[(2-oxocyclopentyl)methyl]-3-[4-(trifluoromethoxy)phenyl]phenyl]propanoate NA 460000 NA NA NA NA TTD
PTGS1 Sodium;2-[3-(4-methylsulfanylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 758000 NA NA NA NA TTD
PTGS1 sodium;2-[4-[[(1R,2S)-2-hydroxycyclopentyl]methyl]-2-(4-hydroxyphenyl)phenyl]propanoate NA 650000 NA NA NA NA TTD
PTGS1 6-Maleimidohexanoic acid NA 800000 NA NA NA NA TTD
PTGS1 2-[1-(4-Chlorobenzoyl)-2-phenylindol-3-yl]acetic acid NA 400000 NA NA NA NA TTD
PTGS1 N-(4-Methoxybenzylidene)-4-sulfamoylaniline NA 313830 NA NA NA NA TTD
PTGS1 Trihydroxychalcone NA 130000 NA NA NA NA TTD
PTGS1 Fenofibric Acid NA 950000 NA NA NA NA PubChem|TTD
PTGS1 Ursolic Acid NA 210000 NA NA NA NA PubChem|TTD
PTGS1 Caffeic Acid NA 400000 NA NA NA NA PubChem|TTD
PTGS1 N-(4-Methylbenzylidene)-4-sulfamoylaniline NA 190470 NA NA NA NA TTD
PTGS1 Romazarit NA 6500000 NA NA NA NA TTD
PTGS1 1-cyclohexyl-5-(4-methylsulfonylphenyl)-3-[(Z)-4-nitrobut-1-enyl]pyrazole NA 1000000 NA NA NA NA TTD
PTGS1 Clobuzarit NA 950000 NA NA NA NA TTD
PTGS1 2-[[2-Amino-2-[1-(3-fluorophenyl)-2-methyl-5-(4-methylsulfonylphenyl)pyrrol-3-yl]acetyl]amino]ethyl nitrate NA 140000 NA NA NA NA TTD
PTGS1 2-amino-2-[1-(3-fluorophenyl)-2-methyl-5-(4-methylsulfonylphenyl)pyrrol-3-yl]-N-(2-hydroxyethyl)acetamide NA 300000 NA NA NA NA TTD
PTGS1 (NZ)-N-[[1-(3,4-difluorophenyl)-2-methyl-5-(4-methylsulfonylphenyl)pyrrol-3-yl]methylidene]hydroxylamine NA 161000 NA NA NA NA TTD
PTGS1 Fangchinoline NA 129000 NA NA NA NA PubChem|TTD
PTGS1 5-Chloro-3-[[1-(4-chlorophenyl)triazol-4-yl]methyl]-1,3-benzoxazol-2-one NA 111340 NA NA NA NA TTD
PTGS1 3-[[1-(4-Chlorophenyl)triazol-4-yl]methyl]-6-methyl-1,3-benzoxazol-2-one NA 389200 NA NA NA NA TTD