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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTGS2 2-(4-methylsulfonylphenyl)-N-(thiophen-2-ylmethyl)pyrimidin-4-amine NA 108000000|108697611 NA NA NA NA BindingDB
PTGS2 2-(4-methylsulfonylphenyl)-4-N-propan-2-yl-6-N-(thiophen-2-ylmethyl)pyrimidine-4,6-diamine NA 97000000|97088994 NA NA NA NA BindingDB
PTGS2 6-N-benzyl-2-(4-methylsulfonylphenyl)-4-N-propan-2-ylpyrimidine-4,6-diamine NA 3650000|3652330 NA NA NA NA BindingDB
PTGS2 4-[4-(Thiophen-3-ylmethylamino)-6-(trifluoromethyl)pyrimidin-2-yl]benzenesulfonamide NA 19200000|19268149 NA NA NA NA BindingDB
PTGS2 2-(4-methylsulfonylphenyl)-N-(thiophen-3-ylmethyl)-6-(trifluoromethyl)pyrimidin-4-amine NA 21500000|21505523 NA NA NA NA BindingDB
PTGS2 NA 20200000|20284299 NA NA NA NA BindingDB
PTGS2 NA 12500000|12594473 NA NA NA NA BindingDB
PTGS2 N-[(3-methylphenyl)methyl]-2-(4-methylsulfonylphenyl)-6-(trifluoromethyl)pyrimidin-4-amine NA 518000|518143 NA NA NA NA BindingDB
PTGS2 N-[(2-methylphenyl)methyl]-2-(4-methylsulfonylphenyl)-6-(trifluoromethyl)pyrimidin-4-amine NA 174000|174828 NA NA NA NA BindingDB
PTGS2 4-[4-(Thiophen-2-ylmethylamino)-6-(trifluoromethyl)pyrimidin-2-yl]benzenesulfonamide NA 6340000|6345268 NA NA NA NA BindingDB
PTGS2 4-[4-(Benzylamino)-6-(trifluoromethyl)pyrimidin-2-yl]benzenesulfonamide NA 300000|300303 NA NA NA NA BindingDB
PTGS2 6-ethylsulfonyl-2-(4-methylsulfonylphenyl)-N-(thiophen-2-ylmethyl)pyrimidin-4-amine NA 6920000|6920540 NA NA NA NA BindingDB
PTGS2 N-benzyl-6-ethylsulfonyl-2-(4-methylsulfonylphenyl)pyrimidin-4-amine NA 11000000|11025543 NA NA NA NA BindingDB
PTGS2 6-ethylsulfanyl-2-(4-methylsulfonylphenyl)-N-(thiophen-2-ylmethyl)pyrimidin-4-amine NA 833000000|833335724 NA NA NA NA BindingDB
PTGS2 N-[(4-fluorophenyl)methyl]-2-(4-methylsulfonylphenyl)-6-(trifluoromethyl)pyrimidin-4-amine NA 12900000|12953586 NA NA NA NA BindingDB
PTGS2 6-chloro-2-(4-methylsulfonylphenyl)-N-(thiophen-2-ylmethyl)pyrimidin-4-amine NA 833000000|833335724 NA NA NA NA BindingDB
PTGS2 N-benzyl-6-ethylsulfanyl-2-(4-methylsulfonylphenyl)pyrimidin-4-amine NA 41400000|41494449|41494448.81 NA NA NA NA BindingDB|TTD
PTGS2 N-benzyl-6-chloro-2-(4-methylsulfonylphenyl)pyrimidin-4-amine NA 91700000|91744492 NA NA NA NA BindingDB
PTGS2 N-[(4-methylphenyl)methyl]-2-(4-methylsulfonylphenyl)-6-(trifluoromethyl)pyrimidin-4-amine NA 20600000|20661412 NA NA NA NA BindingDB
PTGS2 BS3YU156EO NA 400000000|400000008 NA NA NA NA BindingDB