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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTGS2 2-[1-(4-Chlorobenzoyl)-2-ethylindol-3-yl]acetic acid NA 400000 NA NA NA NA TTD
PTGS2 1-(4-chlorophenyl)-5-(4-(methylsulfonyl)phenyl)-1H-tetrazole NA 110000 NA NA NA NA BindingDB|TTD
PTGS2 5-(4-(methylsulfonyl)phenyl)-1-phenyl-1H-tetrazole NA 200000 NA NA NA NA BindingDB|TTD
PTGS2 5-Chloro-2-(4-methylsulfonylcyclohexyl)-3-(3-methylthiophen-1-ium-1-yl)pyran-4-one NA 736037.6 NA NA NA NA BindingDB|TTD
PTGS2 Piroxicam NA 102000|102800|218000 NA NA NA NA BindingDB|GtoPDB|PubChem|TTD
PTGS2 N-[4-[2-(3,4-dichlorophenyl)ethyl]phenyl]-4-hydroxy-1,1-dioxo-2H-1lambda6,2-benzothiazine-3-carboxamide NA 467000 NA NA NA NA BindingDB
PTGS2 N-(3',4'-Dichloro[1,1'-biphenyl]-4-yl)-4-hydroxy-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide NA 263000 NA NA NA NA BindingDB|TTD
PTGS2 Cefepime NA NA NA NA NA 269998 PubChem
PTGS2 Ceftazidime NA NA NA NA NA 300000 PubChem
PTGS2 Sodium;2-[4-[(2-oxocyclopentyl)methyl]-3-phenylphenyl]propanoate NA 290000 NA NA NA NA TTD
PTGS2 Sodium;2-[3-(4-methylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 420000 NA NA NA NA TTD
PTGS2 Disodium;4-[5-(1-carboxylatoethyl)-2-[(2-oxocyclopentyl)methyl]phenyl]benzoate NA 1000000 NA NA NA NA TTD
PTGS2 Sodium;2-[4-[(2-oxocyclopentyl)methyl]-2-[4-(trifluoromethoxy)phenyl]phenyl]propanoate NA 1000000 NA NA NA NA TTD
PTGS2 Sodium;2-[2-iodo-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 540000 NA NA NA NA TTD
PTGS2 Sodium;2-[3-(4-methoxyphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 1000000 NA NA NA NA TTD
PTGS2 Sodium;2-[2-(4-methylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 540000 NA NA NA NA TTD
PTGS2 Sodium;2-[2-(4-methylsulfanylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 150000 NA NA NA NA TTD
PTGS2 Sodium;2-[2-(4-methoxyphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 430000 NA NA NA NA TTD
PTGS2 Sodium;2-[3-(4-methylsulfanylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 1000000 NA NA NA NA TTD
PTGS2 2-[(3Z)-6-fluoro-2-methyl-3-[(3-phenylmethoxyphenyl)methylidene]inden-1-yl]acetic acid NA 286100 NA NA NA NA BindingDB