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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
PTGS2 2-(4-Chlorophenyl)-3-(4-methylsulfonylanilino)-1,3-thiazolidin-4-one NA 121700 NA NA NA NA BindingDB|TTD
PTGS2 p-Terphenyl NA 144000 NA NA NA NA BindingDB|TTD
PTGS2 Romazarit NA 6500000 NA NA NA NA BindingDB|TTD
PTGS2 Clobuzarit NA 950000 NA NA NA NA BindingDB|TTD
PTGS2 N-cyclohex-3-en-1-yl-2-(4-methylsulfonylphenyl)-6-(trifluoromethyl)pyrimidin-4-amine NA 30300000|30395550 NA NA NA NA BindingDB
PTGS2 2-(4-methylsulfonylphenyl)-N-(3-thiophen-2-ylpropyl)-6-(trifluoromethyl)pyrimidin-4-amine NA 826000|826457 NA NA NA NA BindingDB
PTGS2 N-[3-(1-methylpyrrol-2-yl)propyl]-2-(4-methylsulfonylphenyl)-6-(trifluoromethyl)pyrimidin-4-amine NA 251000|251258 NA NA NA NA BindingDB
PTGS2 2-Anilinophenylacetic acid NA 3467369|3467368.5 NA NA NA NA BindingDB|TTD
PTGS2 Cianidanol NA 130000 NA NA NA NA PubChem
PTGS2 2-[2-Iodo-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 540000 NA NA NA NA BindingDB
PTGS2 2-[4-[(2-Oxocyclopentyl)methyl]-3-phenylphenyl]propanoate NA 290000 NA NA NA NA BindingDB
PTGS2 2-[3-(4-Methylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 420000 NA NA NA NA BindingDB
PTGS2 2-[2-(4-Methylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 540000 NA NA NA NA BindingDB
PTGS2 2-[2-(4-Methoxyphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 430000 NA NA NA NA BindingDB
PTGS2 2-[2-(4-Methylsulfanylphenyl)-4-[(2-oxocyclopentyl)methyl]phenyl]propanoate NA 150000 NA NA NA NA BindingDB
PTGS2 Tarenflurbil NA 123000 NA NA NA NA BindingDB|PubChem|TTD
PTGS2 N'-[(E)-(4-oxo-4H-chromen-3-yl)methylidene]benzenecarbohydrazide NA 802320 NA NA NA NA BindingDB|TTD
PTGS2 4-methyl-N''-((4-oxo-4H-chromen-3-yl)methylene)benzenesulfonohydrazide NA 203690 NA NA NA NA BindingDB|TTD
PTGS2 Acetic acid 2-ethylsulfanyl-phenyl ester NA 200000 NA NA NA NA BindingDB|TTD
PTGS2 7,8-dichloro-2-(trifluoromethyl)-2H-chromene-3-carboxylic Acid NA 300000 NA NA NA NA BindingDB|TTD