| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| PTH1R |
Formononetin |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| PTH1R |
Rescinnamine |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
Amentoflavone |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
Sulfaquinoxaline |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
Warfarin |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
Testosterone Propionate |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| PTH1R |
Cinnamaldehyde |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| PTH1R |
Mefloquine Hydrochloride |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| PTH1R |
Gabexate Mesilate |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
2-Cyclohexyl-8-(2-o-tolyl-ethanesulfonyl)-1,3,8-triaza-spiro[4.5]dec-1-en-4-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| PTH1R |
Isoimperatorin |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| PTH1R |
Prazosin Hydrochloride |
NA |
NA |
NA |
NA |
112202 |
NA |
PubChem |
| PTH1R |
(R)-[(2S,5R)-5-ethenyl-1-azabicyclo[2.2.2]octan-2-yl]-(6-methoxyquinolin-4-yl)methanol |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTH1R |
Dibenzazepine |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| PTK2 |
4-(2-methoxyethylamino)-N-(5-(7-methoxyquinolin-4-yloxy)pyridin-2-yl)-2-oxo-1-phenyl-1,2-dihydropyridine-3-carboxamide |
NA |
125000 |
NA |
NA |
NA |
NA |
TTD |
| PTK2 |
4-(Pyridin-3-yl)pyrimidin-2-amine |
NA |
NA |
159000 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| PTK2 |
N-(2-aminophenyl)-6-[(4-ethyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)sulfanyl]hexanamide |
NA |
140640 |
NA |
NA |
NA |
NA |
BindingDB |
| PTK2 |
6-[(4-Prop-2-enyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)sulfanyl]hexanoic acid |
NA |
124300 |
NA |
NA |
NA |
NA |
BindingDB |
| PTK2 |
N-hydroxy-6-[(4-prop-2-enyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)sulfanyl]hexanamide |
NA |
189360 |
NA |
NA |
NA |
NA |
BindingDB |
| PTK2 |
6-[(4-ethyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)sulfanyl]-N-hydroxyhexanamide |
NA |
124030 |
NA |
NA |
NA |
NA |
BindingDB |